# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2408616 | 13f | IC50 | = | 0.014 | uM | ALA2410824 | 7.85 | nM | Homo sapiens | ||
2. | ALA2408616 | 13f | IC50 | = | 0.02 | uM | ALA2410822 | 7.70 | nM | Homo sapiens | ||
3. | ALA2408616 | 13f | ERH | = | 0.39 | ALA2410647 | Mus musculus | |||||
4. | ALA2408616 | 13f | ERH | = | 0.48 | ALA2410646 | Homo sapiens | |||||
5. | ALA2408616 | 13f | Vdss | = | 1 | L/Kg | ALA2410652 | L.kg-1 | Mus musculus | |||
6. | ALA2408616 | 13f | IC50 | = | 1.7 | uM | ALA2410823 | 5.77 | nM | Homo sapiens | ||
7. | ALA2408616 | 13f | t1/2 | = | 1.8 | hr | ALA2410655 | hr | Mus musculus | |||
8. | ALA2408616 | 13f | CL | = | 10 | ml/min.kg | ALA2410656 | mL.min-1.kg-1 | Mus musculus | |||
9. | ALA2408616 | 13f | Cmax | = | 18.6 | uM | ALA2410653 | nM | Mus musculus | |||
10. | ALA2408616 | 13f | INH | > | 50 | % | ALA2410639 | % | Homo sapiens | |||
11. | ALA2408616 | 13f | INH | > | 50 | % | ALA2410638 | % | Homo sapiens | |||
12. | ALA2408616 | 13f | INH | > | 50 | % | ALA2410637 | % | Homo sapiens | |||
13. | ALA2408616 | 13f | INH | > | 50 | % | ALA2410501 | % | Homo sapiens | |||
14. | ALA2408616 | 13f | F | = | 98 | % | ALA2410650 | % | Mus musculus | |||
15. | ALA2408616 | 13f | AUC | = | 3440 | ng.hr/ml | ALA2410654 | ng.hr.mL-1 | Mus musculus | |||
16. | ALA2408616 | 13f | AUC | = | 33710 | ng.hr/ml | ALA2410651 | ng.hr.mL-1 | Mus musculus | |||
17. | ALA2408616 | 13f | IC50 | > | 20 | uM | ALA2410657 | nM | Homo sapiens | |||
18. | ALA2408616 | 13f | AUC | 0 | ALA2410642 | Not Determined | Mus musculus | |||||
19. | ALA2408616 | 13f | F | 0 | ALA2410641 | Not Determined | % | Mus musculus | ||||
20. | ALA2408616 | 13f | Cmax | 0 | ALA2410643 | Not Determined | Mus musculus |