# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2408632 | 4A | IC50 | = | 2.1 | nM | ALA2410614 | 8.68 | nM | Homo sapiens | ||
2. | ALA2408632 | 4A | IC50 | = | 3.7 | nM | ALA2410612 | 8.43 | nM | Mus musculus | ||
3. | ALA2408632 | 4A | logD | = | 1.42 | ALA2410613 | ||||||
4. | ALA2408632 | 4A | IC50 | = | 3528 | nM | ALA2410611 | 5.45 | nM | Homo sapiens | ||
5. | ALA2408632 | 4A | Ratio IC50 | = | 1680 | ALA2410610 | ||||||
6. | ALA2408632 | 4A | Activity | = | 144 | % | ALA2410609 | % | Mus musculus | |||
7. | ALA2408632 | 4A | F | = | 19 | % | ALA2410608 | % | Rattus norvegicus | |||
8. | ALA2408632 | 4A | CL | = | 3 | ml/min.kg | ALA2410607 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA2408632 | 4A | Vdss | = | 0.34 | L/Kg | ALA2410606 | L.kg-1 | Rattus norvegicus | |||
10. | ALA2408632 | 4A | t1/2 | = | 3.7 | hr | ALA2410604 | hr | Rattus norvegicus | |||
11. | ALA2408632 | 4A | AUC/dose | = | 2.4 | microM.hr/mg/kg | ALA2410603 | microM.hr/mg/kg | Rattus norvegicus | |||
12. | ALA2408632 | 4A | Activity | = | 144 | % | ALA4392496 | % | Mus musculus | |||
13. | ALA2408632 | 4A | Ki | = | 5.39 | uM | ALA4392494 | 5.27 | nM | Homo sapiens | ||
14. | ALA2408632 | 4A | logD | = | 1.42 | ALA4392493 | ||||||
15. | ALA2408632 | 4A | IC50 | > | 2000 | nM | ALA4392492 | nM | Homo sapiens | |||
16. | ALA2408632 | 4A | IC50 | = | 2.8 | nM | ALA4392491 | 8.55 | nM | Mus musculus | ||
17. | ALA2408632 | 4A | IC50 | = | 1.5 | nM | ALA4392490 | 8.82 | nM | Homo sapiens |