# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2409730 | 4a, diastereomer 1 | IC50 | = | 1.22 | uM | ALA2412207 | 5.91 | nM | Mus musculus | ||
2. | ALA2409730 | 4a, diastereomer 1 | Drug metabolism | = | 18 | % | ALA2412204 | % | Homo sapiens | |||
3. | ALA2409730 | 4a, diastereomer 1 | Drug metabolism | = | 19 | % | ALA2412203 | % | ||||
4. | ALA2409730 | 4a, diastereomer 1 | IC50 | = | 0.024 | uM | ALA2412206 | 7.62 | nM | Homo sapiens | ||
5. | ALA2409730 | 4a, diastereomer 1 | IC50 | = | 0.031 | uM | ALA2412206 | 7.51 | nM | Homo sapiens | ||
6. | ALA2409730 | 4a, diastereomer 1 | IC50 | = | 0.328 | uM | ALA2412207 | 6.48 | nM | Mus musculus | ||
7. | ALA2409730 | 4a, diastereomer 1 | IC50 | = | 0.246 | uM | ALA2412205 | 6.61 | nM | Rattus norvegicus | ||
8. | ALA2409730 | 4a, diastereomer 1 | Stability | 0 | ALA2412202 | Stable | % | |||||
9. | ALA2409730 | 4a, diastereomer 1 | Stability | 0 | ALA2412200 | Stable | % | |||||
10. | ALA2409730 | 4a, diastereomer 1 | Stability | 0 | ALA2412201 | Stable | % |