# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2415106 | 6a | INH | = | 50.9 | % | ALA2417344 | % | Homo sapiens | |||
2. | ALA2415106 | 6a | INH | = | 82 | % | ALA2417343 | % | Homo sapiens | |||
3. | ALA2415106 | 6a | Imax | = | 83.2 | % | ALA2417345 | % | Homo sapiens | |||
4. | ALA2415106 | 6a | IC50 | = | 10.8 | uM | ALA2416379 | 4.97 | nM | Homo sapiens | ||
5. | ALA2415106 | 6a | IC50 | = | 0.67 | uM | ALA3364117 | 6.17 | nM | Homo sapiens | ||
6. | ALA2415106 | 6a | Efficacy | = | 73 | % | ALA3364118 | % | Homo sapiens | |||
7. | ALA2415106 | 6a | IC50 | = | 4.07 | uM | ALA3364119 | 5.39 | nM | Homo sapiens | ||
8. | ALA2415106 | 6a | Efficacy | = | 83 | % | ALA3364120 | % | Homo sapiens | |||
9. | ALA2415106 | 6a | IC50 | > | 100 | uM | ALA3364121 | nM | Mus musculus | |||
10. | ALA2415106 | 6a | Ki | = | 0.48 | uM | ALA3364122 | 6.32 | nM | Homo sapiens | ||
11. | ALA2415106 | 6a | Ki | = | 4.11 | uM | ALA3364123 | 5.39 | nM | Homo sapiens | ||
12. | ALA2415106 | 6a | Ratio Ki | = | 9 | ALA3364437 | ||||||
13. | ALA2415106 | 6a | IC50 | = | 10.8 | uM | ALA4424992 | 4.97 | nM | Homo sapiens | ||
14. | ALA2415106 | 6a | Efficacy | = | 83.2 | % | ALA4424992 | % | Homo sapiens | |||
15. | ALA2415106 | 6a | IC50 | = | 14.2 | uM | ALA4700533 | 4.85 | nM | Homo sapiens | ||
16. | ALA2415106 | 6a | CC50 | = | 98.4 | uM | ALA4700532 | nM | Homo sapiens | |||
17. | ALA2415106 | 6a | IC50 | = | 155 | nM | ALA4679265 | 6.81 | nM | Homo sapiens | ||
18. | ALA2415106 | 6a | IC50 | = | 41 | nM | ALA4679264 | 7.39 | nM | Rattus norvegicus | ||
19. | ALA2415106 | 6a | IC50 | = | 44 | nM | ALA4679263 | 7.36 | nM | Mus musculus | ||
20. | ALA2415106 | 6a | Cmax | = | 519 | nM | ALA4679262 | nM |