| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2417553 | 44 | IC50 | = | 2 | nM | ALA2423499 | 8.70 | nM | Homo sapiens | ||
| 2. | ALA2417553 | 44 | IC50 | = | 33 | nM | ALA2423498 | 7.48 | nM | Homo sapiens | ||
| 3. | ALA2417553 | 44 | Ratio IC50 | = | 15.1 | ALA2423497 | ||||||
| 4. | ALA2417553 | 44 | Ratio IC50 | > | 50 | ALA2423496 | Homo sapiens | |||||
| 5. | ALA2417553 | 44 | INH | = | 5 | % | ALA2423495 | % | Homo sapiens | |||
| 6. | ALA2417553 | 44 | INH | = | 1 | % | ALA2423313 | % | Homo sapiens | |||
| 7. | ALA2417553 | 44 | IC50 | = | 106 | uM | ALA2423312 | nM | Homo sapiens | |||
| 8. | ALA2417553 | 44 | IC50 | = | 1.1 | uM | ALA2423309 | 5.96 | nM | Homo sapiens | ||
| 9. | ALA2417553 | 44 | Ratio IC50 | = | 550 | ALA2423311 | ||||||
| 10. | ALA2417553 | 44 | IC50 | = | 2440 | nM | ALA2423310 | 5.61 | nM | Rattus norvegicus | ||
| 11. | ALA2417553 | 44 | t1/2 | = | 16 | min | ALA2423500 | hr | Rattus norvegicus | |||
| 12. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423308 | hr | Homo sapiens | |||
| 13. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423307 | hr | Rattus norvegicus | |||
| 14. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423305 | hr | Homo sapiens | |||
| 15. | ALA2417553 | 44 | LC50 | = | 61.4 | uM | ALA2423306 | nM | Homo sapiens | |||
| 16. | ALA2417553 | 44 | Selectivity Index | = | 15.1 | ALA3424483 | ||||||
| 17. | ALA2417553 | 44 | IC50 | = | 2440 | nM | ALA3424482 | 5.61 | nM | Rattus norvegicus | ||
| 18. | ALA2417553 | 44 | IC50 | > | 5000 | nM | ALA3424481 | nM | Homo sapiens | |||
| 19. | ALA2417553 | 44 | IC50 | = | 33 | nM | ALA3424480 | 7.48 | nM | Homo sapiens | ||
| 20. | ALA2417553 | 44 | IC50 | = | 2 | nM | ALA3424479 | 8.70 | nM | Homo sapiens |
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