# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2417553 | 44 | Selectivity Index | = | 15.1 | ALA3424483 | ||||||
2. | ALA2417553 | 44 | IC50 | = | 2440 | nM | ALA3424482 | 5.61 | nM | Rattus norvegicus | ||
3. | ALA2417553 | 44 | IC50 | > | 5000 | nM | ALA3424481 | nM | Homo sapiens | |||
4. | ALA2417553 | 44 | IC50 | = | 33 | nM | ALA3424480 | 7.48 | nM | Homo sapiens | ||
5. | ALA2417553 | 44 | IC50 | = | 2 | nM | ALA3424479 | 8.70 | nM | Homo sapiens | ||
6. | ALA2417553 | 44 | t1/2 | = | 16 | min | ALA4016914 | hr | Rattus norvegicus | |||
7. | ALA2417553 | 44 | IC50 | = | 2 | nM | ALA2423499 | 8.70 | nM | Homo sapiens | ||
8. | ALA2417553 | 44 | IC50 | = | 33 | nM | ALA2423498 | 7.48 | nM | Homo sapiens | ||
9. | ALA2417553 | 44 | Ratio IC50 | = | 15.1 | ALA2423497 | ||||||
10. | ALA2417553 | 44 | Ratio IC50 | > | 50 | ALA2423496 | Homo sapiens | |||||
11. | ALA2417553 | 44 | INH | = | 5 | % | ALA2423495 | % | Homo sapiens | |||
12. | ALA2417553 | 44 | INH | = | 1 | % | ALA2423313 | % | Homo sapiens | |||
13. | ALA2417553 | 44 | IC50 | = | 106 | uM | ALA2423312 | nM | Homo sapiens | |||
14. | ALA2417553 | 44 | IC50 | = | 1.1 | uM | ALA2423309 | 5.96 | nM | Homo sapiens | ||
15. | ALA2417553 | 44 | Ratio IC50 | = | 550 | ALA2423311 | ||||||
16. | ALA2417553 | 44 | IC50 | = | 2440 | nM | ALA2423310 | 5.61 | nM | Rattus norvegicus | ||
17. | ALA2417553 | 44 | t1/2 | = | 16 | min | ALA2423500 | hr | Rattus norvegicus | |||
18. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423308 | hr | Homo sapiens | |||
19. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423307 | hr | Rattus norvegicus | |||
20. | ALA2417553 | 44 | t1/2 | > | 150 | min | ALA2423305 | hr | Homo sapiens |