# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2426277 | 56 | INH | = | 97 | % | ALA3389032 | % | Homo sapiens | |||
2. | ALA2426277 | 56 | INH | = | 92 | % | ALA3389031 | % | Homo sapiens | |||
3. | ALA2426277 | 56 | IC50 | = | 0.002 | uM | ALA3389029 | 8.70 | nM | Homo sapiens | ||
4. | ALA2426277 | 56 | IC50 | = | 7.1 | uM | ALA3389028 | 5.15 | nM | Homo sapiens | ||
5. | ALA2426277 | 56 | Therm_solubility | > | 973 | uM | ALA3389027 | nM | ||||
6. | ALA2426277 | 56 | AUC | = | 13.4 | uM.hr | ALA3389025 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
7. | ALA2426277 | 56 | Cmax | = | 2.7 | uM | ALA3389024 | nM | Mus musculus | |||
8. | ALA2426277 | 56 | logD | = | 3.6 | ALA3389023 | ||||||
9. | ALA2426277 | 56 | IC50 | = | 12 | uM | ALA3389022 | 4.92 | nM | Homo sapiens | ||
10. | ALA2426277 | 56 | IC50 | = | 0.14 | uM | ALA3389021 | 6.85 | nM | Homo sapiens | ||
11. | ALA2426277 | 56 | IC50 | = | 0.019 | uM | ALA3389020 | 7.72 | nM | Homo sapiens | ||
12. | ALA2426277 | 56 | IC50 | = | 0.019 | uM | ALA2427158 | 7.72 | nM | Homo sapiens | ||
13. | ALA2426277 | 56 | IC50 | = | 0.14 | uM | ALA2427714 | 6.85 | nM | Homo sapiens | ||
14. | ALA2426277 | 56 | IC50 | = | 12 | uM | ALA2427713 | 4.92 | nM | Homo sapiens | ||
15. | ALA2426277 | 56 | Ratio IC50 | = | 620 | ALA2427712 | ||||||
16. | ALA2426277 | 56 | logD | = | 4.1 | ALA2427707 | ||||||
17. | ALA2426277 | 56 | t1/2 | = | 188 | min | ALA2427705 | hr |