| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2430727 | 35 | IC50 | = | 0.5 | uM | ALA2432259 | 6.30 | nM | Homo sapiens | ||
| 2. | ALA2430727 | 35 | Ratio IC50 | = | 4 | ALA2432255 | ||||||
| 3. | ALA2430727 | 35 | Ratio IC50 | = | 10 | ALA2432254 | ||||||
| 4. | ALA2430727 | 35 | Ratio IC50 | > | 500 | ALA2432253 | ||||||
| 5. | ALA2430727 | 35 | Ratio IC50 | > | 500 | ALA2432252 | ||||||
| 6. | ALA2430727 | 35 | CLH | = | 1 | ml/min.kg | ALA2432251 | mL.min-1.kg-1 | Homo sapiens | |||
| 7. | ALA2430727 | 35 | CLH | = | 4 | ml/min.kg | ALA2432250 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA2430727 | 35 | PPB | > | 99 | % | ALA2432249 | % | Homo sapiens | |||
| 9. | ALA2430727 | 35 | PPB | = | 99 | % | ALA2432247 | % | Rattus norvegicus | |||
| 10. | ALA2430727 | 35 | permeability | = | 12.1 | ucm/s | ALA2432248 | ucm/s | Canis lupus familiaris | |||
| 11. | ALA2430727 | 35 | permeability | = | 10.3 | ucm/s | ALA2432246 | ucm/s | Canis lupus familiaris | |||
| 12. | ALA2430727 | 35 | Kinetic_solubility | = | 81 | uM | ALA2432244 | nM | ||||
| 13. | ALA2430727 | 35 | INH | 0 | ALA2432245 | Not Active | % | Homo sapiens | ||||
| 14. | ALA2430727 | 35 | INH | 0 | ALA2432243 | Not Active | % | Homo sapiens | ||||
| 15. | ALA2430727 | 35 | INH | 0 | ALA2432242 | Not Active | % | Homo sapiens | ||||
| 16. | ALA2430727 | 35 | INH | 0 | ALA2432240 | Not Active | % | Homo sapiens | ||||
| 17. | ALA2430727 | 35 | INH | 0 | ALA2432241 | Not Active | % | Homo sapiens | ||||
| 18. | ALA2430727 | 35 | CL | = | 60 | ml/min.kg | ALA2432239 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 19. | ALA2430727 | 35 | Vd | = | 1.4 | L/Kg | ALA2432238 | L.kg-1 | Rattus norvegicus | |||
| 20. | ALA2430727 | 35 | Cmax | = | 2.1 | uM | ALA2432237 | nM | Rattus norvegicus |
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