# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2431324 | 1, HOCPCA | pKi | = | 6.89 | ALA4020668 | 6.89 | nM | ||||
2. | ALA2431324 | 1, HOCPCA | Ki | = | 0.13 | uM | ALA4020668 | 6.89 | nM | |||
3. | ALA2431324 | 1, HOCPCA | Ki | = | 1.8 | uM | ALA5099990 | 5.75 | nM | Rattus norvegicus | ||
4. | ALA2431324 | 1, HOCPCA | Ki | = | 0.13 | uM | ALA5099989 | 6.89 | nM | Rattus norvegicus | ||
5. | ALA2431324 | 1, HOCPCA | Ki | = | 0.16 | uM | ALA5099988 | 6.80 | nM | Rattus norvegicus | ||
6. | ALA2431324 | 1, HOCPCA | Stability | = | 16 | months | ALA2432574 | months | ||||
7. | ALA2431324 | 1, HOCPCA | Stability | = | 100 | % | ALA2432573 | % | ||||
8. | ALA2431324 | 1, HOCPCA | Stability | = | 96 | % | ALA2432571 | % | ||||
9. | ALA2431324 | 1, HOCPCA | INH | 0 | ALA2432569 | Dose-dependent effect | % | |||||
10. | ALA2431324 | 1, HOCPCA | IC50 | = | 0.073 | uM | ALA2432569 | 7.14 | nM | |||
11. | ALA2431324 | 1, HOCPCA | pIC50 | = | 7.14 | ALA2432569 | 7.14 | nM | ||||
12. | ALA2431324 | 1, HOCPCA | Ki | = | 0.16 | uM | ALA2432575 | 6.80 | nM | |||
13. | ALA2431324 | 1, HOCPCA | BPR | = | 0.37 | ALA2432566 | ||||||
14. | ALA2431324 | 1, HOCPCA | permeability | 0 | ALA2432565 | impermeable | Canis lupus familiaris | |||||
15. | ALA2431324 | 1, HOCPCA | permeability | 0 | ALA2432564 | impermeable | Canis lupus familiaris | |||||
16. | ALA2431324 | 1, HOCPCA | Stability | = | 88 | % | ALA2432563 | % |