# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2431595 | (R)-2 | F | < | 1 | % | ALA3119302 | % | Rattus norvegicus | |||
2. | ALA2431595 | (R)-2 | F | = | 3.5 | % | ALA3116762 | % | Canis lupus familiaris | |||
3. | ALA2431595 | (R)-2 | Ki | = | 11 | nM | ALA3116761 | 7.96 | nM | Homo sapiens | ||
4. | ALA2431595 | (R)-2 | permeability | < | 15 | nm/s | ALA3119289 | nm/s | Homo sapiens | |||
5. | ALA2431595 | (R)-2 | t1/2 | = | 1.5 | hr | ALA2433495 | hr | Canis lupus familiaris | |||
6. | ALA2431595 | (R)-2 | Vdss | = | 1.5 | L/Kg | ALA2433494 | L.kg-1 | Canis lupus familiaris | |||
7. | ALA2431595 | (R)-2 | F | = | 4 | % | ALA2433493 | % | Canis lupus familiaris | |||
8. | ALA2431595 | (R)-2 | Ki | = | 9.7 | nM | ALA2434648 | 8.01 | nM | Homo sapiens | ||
9. | ALA2431595 | (R)-2 | CL | = | 24 | ml/min.kg | ALA2433496 | mL.min-1.kg-1 | Canis lupus familiaris | |||
10. | ALA2431595 | (R)-2 | 2PT | = | 36 | uM | ALA2433500 | uM | ||||
11. | ALA2431595 | (R)-2 | Ki | = | 6900 | nM | ALA2433498 | 5.16 | nM | Homo sapiens | ||
12. | ALA2431595 | (R)-2 | Ki | = | 7300 | nM | ALA2433499 | 5.14 | nM | Homo sapiens | ||
13. | ALA2431595 | (R)-2 | Ki | > | 5000 | nM | ALA2433497 | nM | Homo sapiens |