# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2436225 | 33 | Ratio | = | 0 | L/min/umol | ALA2437633 | L/min/umol | Homo sapiens | |||
2. | ALA2436225 | 33 | Kinact | = | 0.018 | /min | ALA2437634 | /min | Homo sapiens | |||
3. | ALA2436225 | 33 | IC50 | = | 0.022 | uM | ALA2437637 | 7.66 | nM | Homo sapiens | ||
4. | ALA2436225 | 33 | Fu | = | 0.08 | % | ALA2439933 | |||||
5. | ALA2436225 | 33 | Fu | = | 2.8 | % | ALA2439932 | |||||
6. | ALA2436225 | 33 | Tmax | = | 4 | hr | ALA2439934 | hr | Mus musculus | |||
7. | ALA2436225 | 33 | F | = | 8 | % | ALA2439935 | % | Mus musculus | |||
8. | ALA2436225 | 33 | IC20 | > | 10 | uM | ALA2439936 | uM | Homo sapiens | |||
9. | ALA2436225 | 33 | IC50 | = | 18 | uM | ALA2437635 | 4.75 | nM | Homo sapiens | ||
10. | ALA2436225 | 33 | IC50 | > | 20 | uM | ALA2439936 | nM | Homo sapiens | |||
11. | ALA2436225 | 33 | IC50 | = | 23.2 | uM | ALA2437636 | 4.63 | nM | Homo sapiens | ||
12. | ALA2436225 | 33 | Ki | = | 50 | uM | ALA2437634 | 4.30 | nM | Homo sapiens | ||
13. | ALA2436225 | 33 | IC50 | > | 50 | uM | ALA2439942 | nM | Homo sapiens | |||
14. | ALA2436225 | 33 | IC50 | > | 50 | uM | ALA2439941 | nM | Homo sapiens | |||
15. | ALA2436225 | 33 | Cmax | = | 873 | ng/ml | ALA2439938 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
16. | ALA2436225 | 33 | AUC | = | 5980 | ng.hr/ml | ALA2439937 | ng.hr.mL-1 | Mus musculus | |||
17. | ALA2436225 | 33 | Stability | 0 | ALA2439939 | Stable | % | Homo sapiens |