# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441089 | 19 | IC50 | = | 1.6 | nM | ALA2446442 | 8.80 | nM | Rattus norvegicus | ||
2. | ALA2441089 | 19 | IC50 | = | 38 | nM | ALA2446441 | 7.42 | nM | Rattus norvegicus | ||
3. | ALA2441089 | 19 | INH | = | 88 | % | ALA2446440 | % | Rattus norvegicus | |||
4. | ALA2441089 | 19 | INH | = | 78 | % | ALA2446439 | % | Rattus norvegicus | |||
5. | ALA2441089 | 19 | INH | = | 45 | % | ALA2446438 | % | Rattus norvegicus | |||
6. | ALA2441089 | 19 | Activity | = | 29 | % | ALA2446436 | % | marmosets | |||
7. | ALA2441089 | 19 | Activity | = | 44 | % | ALA2446435 | % | marmosets | |||
8. | ALA2441089 | 19 | Activity | = | 3 | % | ALA2446434 | % | marmosets | |||
9. | ALA2441089 | 19 | Activity | = | 29 | % | ALA2446433 | % | marmosets | |||
10. | ALA2441089 | 19 | Drug uptake | = | 1045 | ng/g | ALA2446432 | ng/g | ||||
11. | ALA2441089 | 19 | Kp | = | 66 | ALA2446431 |