# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441831 | 2b, more active atropisomer | Ki | = | 11 | nM | ALA2444439 | 7.96 | nM | Homo sapiens | ||
2. | ALA2441831 | 2b, more active atropisomer | Ki | = | 5.5 | nM | ALA2444440 | 8.26 | nM | Homo sapiens | ||
3. | ALA2441831 | 2b, more active atropisomer | Ki | = | 1.2 | nM | ALA2444438 | 8.92 | nM | Homo sapiens | ||
4. | ALA2441831 | 2b, more active atropisomer | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
5. | ALA2441831 | 2b, more active atropisomer | IC50 | = | 11 | uM | ALA2444436 | 4.96 | nM | Homo sapiens | ||
6. | ALA2441831 | 2b, more active atropisomer | Stability | = | 72 | % | ALA2444178 | % | Mus musculus |