# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441834 | 2d, More active atropisomer | Ki | = | 2.6 | nM | ALA2444439 | 8.59 | nM | Homo sapiens | ||
2. | ALA2441834 | 2d, More active atropisomer | Ki | = | 8.9 | nM | ALA2444440 | 8.05 | nM | Homo sapiens | ||
3. | ALA2441834 | 2d, More active atropisomer | Ki | = | 7.3 | nM | ALA2444438 | 8.14 | nM | Homo sapiens | ||
4. | ALA2441834 | 2d, More active atropisomer | INH | = | 37 | % | ALA2444437 | % | Homo sapiens | |||
5. | ALA2441834 | 2d, More active atropisomer | IC50 | = | 7.7 | uM | ALA2444436 | 5.11 | nM | Homo sapiens | ||
6. | ALA2441834 | 2d, More active atropisomer | Stability | = | 94 | % | ALA2444178 | % | Mus musculus |