# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441836 | 1e, BMS-744891 | Ki | = | 8.3 | nM | ALA2444439 | 8.08 | nM | Homo sapiens | ||
2. | ALA2441836 | 1e, BMS-744891 | Ki | = | 6 | nM | ALA2444439 | 8.22 | nM | Homo sapiens | ||
3. | ALA2441836 | 1e, BMS-744891 | Ki | = | 160 | nM | ALA2444439 | 6.80 | nM | Homo sapiens | ||
4. | ALA2441836 | 1e, BMS-744891 | Ki | = | 7.1 | nM | ALA2444440 | 8.15 | nM | Homo sapiens | ||
5. | ALA2441836 | 1e, BMS-744891 | Ki | = | 5.4 | nM | ALA2444440 | 8.27 | nM | Homo sapiens | ||
6. | ALA2441836 | 1e, BMS-744891 | Ki | > | 30 | nM | ALA2444440 | nM | Homo sapiens | |||
7. | ALA2441836 | 1e, BMS-744891 | Ki | = | 4.6 | nM | ALA2444438 | 8.34 | nM | Homo sapiens | ||
8. | ALA2441836 | 1e, BMS-744891 | Ki | = | 1.9 | nM | ALA2444438 | 8.72 | nM | Homo sapiens | ||
9. | ALA2441836 | 1e, BMS-744891 | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
10. | ALA2441836 | 1e, BMS-744891 | INH | = | 10 | % | ALA2444437 | % | Homo sapiens | |||
11. | ALA2441836 | 1e, BMS-744891 | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
12. | ALA2441836 | 1e, BMS-744891 | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
13. | ALA2441836 | 1e, BMS-744891 | IC50 | = | 23 | uM | ALA2444436 | 4.64 | nM | Homo sapiens | ||
14. | ALA2441836 | 1e, BMS-744891 | IC50 | = | 29 | uM | ALA2444436 | 4.54 | nM | Homo sapiens | ||
15. | ALA2441836 | 1e, BMS-744891 | IC50 | = | 14 | uM | ALA2444436 | 4.85 | nM | Homo sapiens | ||
16. | ALA2441836 | 1e, BMS-744891 | Stability | = | 74 | % | ALA2444178 | % | Mus musculus | |||
17. | ALA2441836 | 1e, BMS-744891 | Stability | = | 65 | % | ALA2444178 | % | Mus musculus | |||
18. | ALA2441836 | 1e, BMS-744891 | Stability | = | 69 | % | ALA2444178 | % | Mus musculus |