# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441837 | 2g, More active atropisomer | Ki | = | 7.4 | nM | ALA2444439 | 8.13 | nM | Homo sapiens | ||
2. | ALA2441837 | 2g, More active atropisomer | Ki | = | 31 | nM | ALA2444439 | 7.51 | nM | Homo sapiens | ||
3. | ALA2441837 | 2g, More active atropisomer | Ki | = | 1.7 | nM | ALA2444440 | 8.77 | nM | Homo sapiens | ||
4. | ALA2441837 | 2g, More active atropisomer | Ki | > | 30 | nM | ALA2444440 | nM | Homo sapiens | |||
5. | ALA2441837 | 2g, More active atropisomer | Ki | = | 2.3 | nM | ALA2444438 | 8.64 | nM | Homo sapiens | ||
6. | ALA2441837 | 2g, More active atropisomer | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
7. | ALA2441837 | 2g, More active atropisomer | INH | = | 11 | % | ALA2444437 | % | Homo sapiens | |||
8. | ALA2441837 | 2g, More active atropisomer | INH | = | 8 | % | ALA2444437 | % | Homo sapiens | |||
9. | ALA2441837 | 2g, More active atropisomer | IC50 | = | 13 | uM | ALA2444436 | 4.89 | nM | Homo sapiens | ||
10. | ALA2441837 | 2g, More active atropisomer | IC50 | = | 13 | uM | ALA2444436 | 4.89 | nM | Homo sapiens | ||
11. | ALA2441837 | 2g, More active atropisomer | Stability | = | 43 | % | ALA2444178 | % | Mus musculus | |||
12. | ALA2441837 | 2g, More active atropisomer | Stability | = | 24 | % | ALA2444178 | % | Mus musculus |