# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441838 | 2h, More active atropisomer | Ki | = | 2.7 | nM | ALA2444439 | 8.57 | nM | Homo sapiens | ||
2. | ALA2441838 | 2h, More active atropisomer | Ki | = | 3.9 | nM | ALA2444440 | 8.41 | nM | Homo sapiens | ||
3. | ALA2441838 | 2h, More active atropisomer | Ki | = | 3.1 | nM | ALA2444438 | 8.51 | nM | Homo sapiens | ||
4. | ALA2441838 | 2h, More active atropisomer | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
5. | ALA2441838 | 2h, More active atropisomer | IC50 | = | 14 | uM | ALA2444436 | 4.85 | nM | Homo sapiens | ||
6. | ALA2441838 | 2h, More active atropisomer | Stability | = | 37 | % | ALA2444178 | % | Mus musculus |