# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441840 | 2j, More active atropisomer | Ki | = | 7.5 | nM | ALA2444439 | 8.12 | nM | Homo sapiens | ||
2. | ALA2441840 | 2j, More active atropisomer | Ki | > | 30 | nM | ALA2444440 | nM | Homo sapiens | |||
3. | ALA2441840 | 2j, More active atropisomer | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
4. | ALA2441840 | 2j, More active atropisomer | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
5. | ALA2441840 | 2j, More active atropisomer | IC50 | = | 40 | uM | ALA2444436 | 4.40 | nM | Homo sapiens | ||
6. | ALA2441840 | 2j, More active atropisomer | Stability | = | 100 | % | ALA2444178 | % | Mus musculus |