| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2441841 | 2k, More active atropisomer | Ratio Ki | = | 9500 | ALA2444177 | ||||||
| 2. | ALA2441841 | 2k, More active atropisomer | Ratio Ki | = | 7250 | ALA2444176 | ||||||
| 3. | ALA2441841 | 2k, More active atropisomer | Ki | = | 0.4 | nM | ALA2444439 | 9.40 | nM | Homo sapiens | ||
| 4. | ALA2441841 | 2k, More active atropisomer | Ki | = | 3.8 | nM | ALA2444440 | 8.42 | nM | Homo sapiens | ||
| 5. | ALA2441841 | 2k, More active atropisomer | Ki | = | 2.9 | nM | ALA2444438 | 8.54 | nM | Homo sapiens | ||
| 6. | ALA2441841 | 2k, More active atropisomer | INH | 0 | ALA2444437 | Not Determined | % | Homo sapiens | ||||
| 7. | ALA2441841 | 2k, More active atropisomer | IC50 | = | 3 | uM | ALA2444436 | 5.52 | nM | Homo sapiens | ||
| 8. | ALA2441841 | 2k, More active atropisomer | Stability | = | 36 | % | ALA2444178 | % | Mus musculus |
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