# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2443026 | 38 | Kd | = | 0.057 | nM | ALA3705819 | 10.24 | 292746 | nM | Homo sapiens | |
2. | ALA2443026 | 38 | DC50 | = | 0.013 | uM | ALA2445179 | uM | Homo sapiens | |||
3. | ALA2443026 | 38 | Kd | = | 0.057 | nM | ALA2445179 | 10.24 | nM | Homo sapiens | ||
4. | ALA2443026 | 38 | IC50 | = | 0.028 | uM | ALA2445178 | 7.55 | nM | Homo sapiens | ||
5. | ALA2443026 | 38 | IC50 | = | 0.011 | uM | ALA2445177 | 7.96 | nM | Homo sapiens | ||
6. | ALA2443026 | 38 | solubility | = | 105 | uM | ALA2445176 | nM | ||||
7. | ALA2443026 | 38 | AUC | = | 7.6 | uM.hr | ALA2445175 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
8. | ALA2443026 | 38 | CL | = | 29.35 | ml/min.kg | ALA2444303 | mL.min-1.kg-1 | Mus musculus | |||
9. | ALA2443026 | 38 | Vdss | = | 4.94 | L/Kg | ALA2444302 | L.kg-1 | Mus musculus | |||
10. | ALA2443026 | 38 | t1/2 | = | 5.46 | hr | ALA2444301 | hr | Mus musculus | |||
11. | ALA2443026 | 38 | TGI | = | 93 | % | ALA2444300 | % | Homo sapiens | |||
12. | ALA2443026 | 38 | TGI | = | 53 | % | ALA2444296 | % | Homo sapiens | |||
13. | ALA2443026 | 38 | TGI | = | 72 | % | ALA2444295 | % | Homo sapiens | |||
14. | ALA2443026 | 38 | Activity | = | 23.4 | % | ALA2444294 | % | Mus musculus | |||
15. | ALA2443026 | 38 | Activity | = | 12.3 | % | ALA2444030 | % | Mus musculus | |||
16. | ALA2443026 | 38 | Activity | = | 19.1 | % | ALA2445181 | % | Mus musculus | |||
17. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444023 | nM | Homo sapiens | |||
18. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
19. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444021 | nM | Homo sapiens | |||
20. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444020 | nM | Homo sapiens |