# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2443139 | 31 | Kd | = | 0.218 | nM | ALA3705819 | 9.66 | 292749 | nM | Homo sapiens | |
2. | ALA2443139 | 31 | DC50 | = | 0.013 | uM | ALA2445179 | uM | Homo sapiens | |||
3. | ALA2443139 | 31 | Kd | = | 0.22 | nM | ALA2445179 | 9.66 | nM | Homo sapiens | ||
4. | ALA2443139 | 31 | IC50 | = | 0.065 | uM | ALA2445178 | 7.19 | nM | Homo sapiens | ||
5. | ALA2443139 | 31 | IC50 | = | 0.074 | uM | ALA2445177 | 7.13 | nM | Homo sapiens | ||
6. | ALA2443139 | 31 | solubility | = | 158 | uM | ALA2445176 | nM | ||||
7. | ALA2443139 | 31 | AUC | = | 4.8 | uM.hr | ALA2445175 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
8. | ALA2443139 | 31 | CL | = | 64.8 | ml/min.kg | ALA2444303 | mL.min-1.kg-1 | Mus musculus | |||
9. | ALA2443139 | 31 | Vdss | = | 18.37 | L/Kg | ALA2444302 | L.kg-1 | Mus musculus | |||
10. | ALA2443139 | 31 | t1/2 | = | 5.44 | hr | ALA2444301 | hr | Mus musculus | |||
11. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444023 | nM | Homo sapiens | |||
12. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444022 | nM | Homo sapiens | |||
13. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444021 | nM | Homo sapiens | |||
14. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444020 | nM | Homo sapiens | |||
15. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444019 | nM | Homo sapiens | |||
16. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444018 | nM | Homo sapiens | |||
17. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444016 | nM | Homo sapiens | |||
18. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444017 | nM | Homo sapiens | |||
19. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444015 | nM | Homo sapiens | |||
20. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444013 | nM | Homo sapiens |