| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3084389 | 36j | Cp | = | 1.4 | uM | ALA1781125 | uM | Mus musculus | |||
| 2. | ALA3084389 | 36j | Cp | = | 0.8 | uM | ALA1781124 | uM | Mus musculus | |||
| 3. | ALA3084389 | 36j | Cp | = | 0.4 | uM | ALA1781123 | uM | Mus musculus | |||
| 4. | ALA3084389 | 36j | INH | = | 39 | % | ALA1781122 | % | Mus musculus | |||
| 5. | ALA3084389 | 36j | INH | = | 30 | % | ALA1781121 | % | Mus musculus | |||
| 6. | ALA3084389 | 36j | INH | = | 28 | % | ALA1781120 | % | Mus musculus | |||
| 7. | ALA3084389 | 36j | Tmax | = | 4.5 | hr | ALA1781118 | hr | Macaca mulatta | |||
| 8. | ALA3084389 | 36j | Cmax | = | 997 | nM | ALA1781117 | nM | Macaca mulatta | |||
| 9. | ALA3084389 | 36j | AUC | = | 16548 | nM/hr | ALA1781116 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca mulatta | ||
| 10. | ALA3084389 | 36j | INH | = | 9 | % | ALA1781114 | % | Homo sapiens | |||
| 11. | ALA3084389 | 36j | INH | = | 0.09 | % | ALA1781113 | % | Homo sapiens | |||
| 12. | ALA3084389 | 36j | AUC | = | 2170 | nM/hr | ALA1781109 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 13. | ALA3084389 | 36j | Cp | = | 275 | nM | ALA1781108 | nM | Mus musculus | |||
| 14. | ALA3084389 | 36j | Activity | = | 91 | % | ALA1781107 | % | Mus musculus | |||
| 15. | ALA3084389 | 36j | Activity | = | 110 | % | ALA1781106 | % | Mus musculus | |||
| 16. | ALA3084389 | 36j | EC50 | = | 140 | nM | ALA1781105 | 6.85 | nM | Mus musculus | ||
| 17. | ALA3084389 | 36j | Activity | = | 96 | % | ALA1781104 | % | Homo sapiens | |||
| 18. | ALA3084389 | 36j | EC50 | = | 3 | nM | ALA1781103 | 8.52 | nM | Homo sapiens | ||
| 19. | ALA3084389 | 36j | IC50 | > | 20 | uM | ALA1781112 | nM | Homo sapiens | |||
| 20. | ALA3084389 | 36j | IC50 | > | 20 | uM | ALA1781111 | nM | Homo sapiens |
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