# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3086086 | 1 | IC50 | = | 9.7 | nM | ALA3088429 | 8.01 | nM | Homo sapiens | ||
2. | ALA3086086 | 1 | Ratio | = | 24.8 | ALA3088428 | Homo sapiens | |||||
3. | ALA3086086 | 1 | Ratio | = | 13.1 | ALA3088427 | Rattus norvegicus | |||||
4. | ALA3086086 | 1 | CLH | = | 127 | microL/min/mg | ALA3088426 | mL.min-1.g-1 | Homo sapiens | |||
5. | ALA3086086 | 1 | CLH | = | 297 | microL/min/mg | ALA3088424 | mL.min-1.g-1 | Rattus norvegicus | |||
6. | ALA3086086 | 1 | Papp | = | 18.1 | ucm/s | ALA3088425 | ucm/s | Sus scrofa | |||
7. | ALA3086086 | 1 | Activity | 0 | ALA3088422 | Active | Homo sapiens | |||||
8. | ALA3086086 | 1 | Activity | 0 | ALA3088423 | Active | Homo sapiens | |||||
9. | ALA3086086 | 1 | CL | = | 3.9 | L/hr/kg | ALA3089610 | mL.min-1.kg-1 | Rattus norvegicus | |||
10. | ALA3086086 | 1 | Vdss | = | 2.52 | L/Kg | ALA3089607 | L.kg-1 | Rattus norvegicus | |||
11. | ALA3086086 | 1 | AUC | = | 0.58 | uM.hr | ALA3089604 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
12. | ALA3086086 | 1 | t1/2 | = | 0.81 | hr | ALA3089600 | hr | Rattus norvegicus |