# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3104879 | 22 | EC50 | = | 0.016 | uM | ALA3107227 | 7.80 | nM | Homo sapiens | ||
2. | ALA3104879 | 22 | CLH | = | 84 | microL/min/mg | ALA3107225 | mL.min-1.g-1 | Rattus norvegicus | |||
3. | ALA3104879 | 22 | EC50 | = | 0.073 | uM | ALA3107223 | 7.14 | nM | Macaca fascicularis | ||
4. | ALA3104879 | 22 | Efficacy | = | 102 | % | ALA3107222 | % | Macaca fascicularis | |||
5. | ALA3104879 | 22 | CLH | = | 29 | microL/min/mg | ALA3107124 | mL.min-1.g-1 | Homo sapiens | |||
6. | ALA3104879 | 22 | Stability | = | 88 | % | ALA3107123 | % | Homo sapiens | |||
7. | ALA3104879 | 22 | CL | = | 0.71 | L/hr/kg | ALA3106572 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA3104879 | 22 | t1/2 | = | 1.5 | hr | ALA3106571 | hr | Rattus norvegicus | |||
9. | ALA3104879 | 22 | Vdss | = | 1.5 | L/Kg | ALA3106570 | L.kg-1 | Rattus norvegicus | |||
10. | ALA3104879 | 22 | F | = | 95 | % | ALA3106569 | % | Rattus norvegicus | |||
11. | ALA3104879 | 22 | CL | = | 0.45 | L/hr/kg | ALA3106568 | mL.min-1.kg-1 | Macaca fascicularis | |||
12. | ALA3104879 | 22 | t1/2 | = | 5.6 | hr | ALA3106567 | hr | Macaca fascicularis | |||
13. | ALA3104879 | 22 | Vdss | = | 1.1 | L/Kg | ALA3106566 | L.kg-1 | Macaca fascicularis | |||
14. | ALA3104879 | 22 | F | = | 29 | % | ALA3106565 | % | Macaca fascicularis | |||
15. | ALA3104879 | 22 | Activity | 0 | ALA3106564 | Not Active | Homo sapiens | |||||
16. | ALA3104879 | 22 | INH | 0 | ALA3106562 | Not Active | % | |||||
17. | ALA3104879 | 22 | IC50 | > | 30 | uM | ALA3106563 | nM | Homo sapiens | |||
18. | ALA3104879 | 22 | Activity | 0 | ALA3106560 | Not Active | Homo sapiens | |||||
19. | ALA3104879 | 22 | PPB | > | 99 | % | ALA3106561 | % | ||||
20. | ALA3104879 | 22 | PPB | > | 99 | % | ALA3106559 | % |