| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3105479 | 85 | EC50 | = | 7 | nM | ALA3108092 | 8.15 | nM | Homo sapiens | ||
| 2. | ALA3105479 | 85 | EC50 | = | 2880 | nM | ALA3108091 | 5.54 | nM | Homo sapiens | ||
| 3. | ALA3105479 | 85 | Activity | 0 | ALA3108086 | Active | Rattus norvegicus | |||||
| 4. | ALA3105479 | 85 | Activity | 0 | ALA3108085 | Dose-dependent effect | Rattus norvegicus | |||||
| 5. | ALA3105479 | 85 | Activity | 0 | ALA3108084 | Active | Rattus norvegicus | |||||
| 6. | ALA3105479 | 85 | Activity | 0 | ALA3108083 | Active | Rattus norvegicus | |||||
| 7. | ALA3105479 | 85 | F | = | 97 | % | ALA3108082 | % | Rattus norvegicus | |||
| 8. | ALA3105479 | 85 | F | = | 62 | % | ALA3108081 | % | Canis lupus familiaris | |||
| 9. | ALA3105479 | 85 | Cmax | = | 4000 | ng/ml | ALA3108080 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 10. | ALA3105479 | 85 | Cmax | = | 3160 | ng/ml | ALA3108079 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
| 11. | ALA3105479 | 85 | Tmax | = | 2 | hr | ALA3108078 | hr | Rattus norvegicus | |||
| 12. | ALA3105479 | 85 | Tmax | = | 2 | hr | ALA3108077 | hr | Canis lupus familiaris | |||
| 13. | ALA3105479 | 85 | AUC | = | 40800 | ng.hr/ml | ALA3108076 | ng.hr.mL-1 | Rattus norvegicus | |||
| 14. | ALA3105479 | 85 | AUC | = | 39300 | ng.hr/ml | ALA3108074 | ng.hr.mL-1 | Canis lupus familiaris | |||
| 15. | ALA3105479 | 85 | t1/2 | = | 4.9 | hr | ALA3108075 | hr | Rattus norvegicus | |||
| 16. | ALA3105479 | 85 | t1/2 | = | 6.9 | hr | ALA3108073 | hr | Canis lupus familiaris | |||
| 17. | ALA3105479 | 85 | CL | = | 4 | ml/min.Kg | ALA3108072 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 18. | ALA3105479 | 85 | CL | = | 0.8 | ml/min.Kg | ALA3108070 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 19. | ALA3105479 | 85 | Vdss | = | 1.6 | L/Kg | ALA3108071 | L.kg-1 | Rattus norvegicus | |||
| 20. | ALA3105479 | 85 | Vdss | = | 0.45 | L/Kg | ALA3106639 | L.kg-1 | Canis lupus familiaris |
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