# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3108870 | 42 | pIC50 | = | 2.23 | ALA4480801 | nM | |||||
2. | ALA3108870 | 42 | pIC50 | = | 2.23 | ALA4480800 | nM | |||||
3. | ALA3108870 | 42 | IC50 | = | 0.015 | uM | ALA3110581 | 7.82 | nM | Trypanosoma brucei | ||
4. | ALA3108870 | 42 | INH | > | 80 | % | ALA3110580 | % | Trypanosoma brucei | |||
5. | ALA3108870 | 42 | IC50 | = | 0.172 | uM | ALA3110579 | 6.76 | nM | Trypanosoma cruzi | ||
6. | ALA3108870 | 42 | INH | > | 80 | % | ALA3110578 | % | Trypanosoma cruzi | |||
7. | ALA3108870 | 42 | Ki | = | 52 | nM | ALA3110577 | 7.28 | nM | Trypanosoma brucei | ||
8. | ALA3108870 | 42 | Ki | = | 240 | nM | ALA3110576 | 6.62 | nM | Trypanosoma brucei | ||
9. | ALA3108870 | 42 | INH | 0 | ALA3110575 | Not Active | % | Oryctolagus cuniculus | ||||
10. | ALA3108870 | 42 | Activity | 0 | ALA3110652 | Not Active | Trypanosoma brucei brucei | |||||
11. | ALA3108870 | 42 | ED50 | = | 46 | uM | ALA3110651 | uM | Homo sapiens | |||
12. | ALA3108870 | 42 | Kinetic_solubility | > | 81 | ug ml-1 | ALA3110650 | ug.mL-1 | ||||
13. | ALA3108870 | 42 | t1/2 | 0 | ALA3110649 | Not Determined | ||||||
14. | ALA3108870 | 42 | t1/2 | > | 30 | min | ALA3110648 | hr | Rattus norvegicus | |||
15. | ALA3108870 | 42 | t1/2 | 0 | ALA3110647 | Not Determined | Homo sapiens | |||||
16. | ALA3108870 | 42 | Stability | > | 95 | % | ALA3110646 | % | Mus musculus | |||
17. | ALA3108870 | 42 | Stability | > | 95 | % | ALA3110645 | % | Homo sapiens |