| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Activity | 0 | ALA3110751 | Not Active | Trypanosoma brucei brucei | |||||
| 2. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Activity | 0 | ALA3110758 | Active | Trypanosoma brucei brucei | |||||
| 3. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Cmax | = | 3998 | nM | ALA3110740 | nM | Mus musculus | |||
| 4. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Cmax | = | 9167 | nM | ALA3110739 | nM | Mus musculus | |||
| 5. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Drug metabolism | 0 | ALA3110760 | Not Active | Homo sapiens | |||||
| 6. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Drug metabolism | 0 | ALA3110759 | Not Active | Homo sapiens | |||||
| 7. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Fu | = | 100 | % | ALA3110742 | Homo sapiens | ||||
| 8. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 0.17 | uM | ALA3110905 | 6.77 | nM | Trypanosoma brucei brucei | ||
| 9. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 2.13 | uM | ALA3110754 | 5.67 | nM | Homo sapiens | ||
| 10. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 2.44 | uM | ALA3110755 | 5.61 | nM | Homo sapiens | ||
| 11. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 5.46 | uM | ALA3110763 | 5.26 | nM | Mus musculus | ||
| 12. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 170 | nM | ALA3110752 | 6.77 | nM | Trypanosoma brucei | ||
| 13. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | IC50 | = | 176 | nM | ALA3110753 | 6.75 | nM | Trypanosoma brucei | ||
| 14. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Ki | = | 0.96 | uM | ALA3110901 | 6.02 | nM | |||
| 15. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Papp | = | 1.4 | ucm/s | ALA3110747 | ucm/s | Homo sapiens | |||
| 16. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Papp | = | 3 | ucm/s | ALA3110749 | ucm/s | Homo sapiens | |||
| 17. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Papp | = | 102 | % | ALA3110748 | % | Homo sapiens | |||
| 18. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Papp | = | 104 | % | ALA3110746 | % | Homo sapiens | |||
| 19. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Ratio | = | 0.5 | ALA3110744 | Homo sapiens | |||||
| 20. | ALA3110070 | 1b, 2-fluoro-3'-deoxyadenosine, 2-fluorocordycepin | Stability | = | 98 | % | ALA3110750 | % | Homo sapiens |
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