# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3115061 | 38 | IC50 | = | 0.004 | uM | ALA3116955 | 8.40 | nM | Homo sapiens | ||
2. | ALA3115061 | 38 | IC50 | = | 33 | nM | ALA3116954 | 7.48 | nM | Homo sapiens | ||
3. | ALA3115061 | 38 | IC50 | = | 74 | nM | ALA3116953 | 7.13 | nM | Homo sapiens | ||
4. | ALA3115061 | 38 | logD | = | 0.05 | ALA3116952 | ||||||
5. | ALA3115061 | 38 | solubility | = | 1.54 | mg/ml | ALA3116951 | ug.mL-1 | ||||
6. | ALA3115061 | 38 | Drug metabolism | = | 3 | % | ALA3116950 | % | Homo sapiens | |||
7. | ALA3115061 | 38 | Drug metabolism | = | 0 | % | ALA3116949 | % | Rattus norvegicus | |||
8. | ALA3115061 | 38 | Drug metabolism | = | 0 | % | ALA3116947 | % | ||||
9. | ALA3115061 | 38 | Stability | 0 | ALA3116948 | Stable | % | Homo sapiens | ||||
10. | ALA3115061 | 38 | Stability | 0 | ALA3116946 | Stable | % | Mus musculus | ||||
11. | ALA3115061 | 38 | Stability | 0 | ALA3116945 | Stable | % | Rattus norvegicus | ||||
12. | ALA3115061 | 38 | permeability | = | 1 | 10'-7 cm/s | ALA3116944 | 10'-7 cm/s | Homo sapiens | |||
13. | ALA3115061 | 38 | IC50 | > | 30 | uM | ALA3116943 | nM | Homo sapiens | |||
14. | ALA3115061 | 38 | Activity | < | 10 | % | ALA3116942 | % | Homo sapiens | |||
15. | ALA3115061 | 38 | Activity | < | 10 | % | ALA3116941 | % | Homo sapiens | |||
16. | ALA3115061 | 38 | Activity | < | 10 | % | ALA3116940 | % | Homo sapiens | |||
17. | ALA3115061 | 38 | IC50 | > | 10 | uM | ALA3116939 | nM | Homo sapiens | |||
18. | ALA3115061 | 38 | t1/2 | = | 0.24 | hr | ALA3116938 | hr | Rattus norvegicus | |||
19. | ALA3115061 | 38 | C0 | = | 1.7 | ug ml-1 | ALA3116937 | ug ml-1 | Rattus norvegicus | |||
20. | ALA3115061 | 38 | Vdss | = | 3.6 | L/Kg | ALA3116936 | L.kg-1 | Rattus norvegicus |