Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Assay	Assay Organism
1.	ALA3121095	R,S(+)-4a, R,S-4a	IC50	>	30	uM	ALA3123344		nM	Homo sapiens
2.	ALA3121095	R,S(+)-4a, R,S-4a	IC50	>	30	uM	ALA3123346		nM	Homo sapiens
3.	ALA3121095	R,S(+)-4a, R,S-4a	Ki	=	3.8	nM	ALA3123356	8.42	nM	Homo sapiens
4.	ALA3121095	R,S(+)-4a, R,S-4a	Ki	=	7.3	nM	ALA3123355	8.14	nM	Rattus norvegicus
5.	ALA3121095	R,S(+)-4a, R,S-4a	t1/2	>	40	min	ALA3123341		hr
6.	ALA3121095	R,S(+)-4a, R,S-4a	t1/2	>	40	min	ALA3123339		hr	Rattus norvegicus
7.	ALA3121095	R,S(+)-4a, R,S-4a	t1/2	>	40	min	ALA3123340		hr	Canis lupus familiaris
8.	ALA3121095	R,S(+)-4a, R,S-4a	t1/2	>	40	min	ALA3123338		hr
9.	ALA3121095	R,S(+)-4a, R,S-4a	t1/2	>	40	min	ALA3123337		hr	Homo sapiens
10.	ALA3121095	R,S(+)-4a, R,S-4a	INH	<	10	%	ALA3123335		%	Homo sapiens
11.	ALA3121095	R,S(+)-4a, R,S-4a	INH	<	10	%	ALA3123336		%	Homo sapiens
12.	ALA3121095	R,S(+)-4a, R,S-4a	INH	<	10	%	ALA3123334		%	Homo sapiens
13.	ALA3121095	R,S(+)-4a, R,S-4a	IC50	=	14	uM	ALA3123331	4.85	nM	Homo sapiens
14.	ALA3121095	R,S(+)-4a, R,S-4a	Papp	=	16.4	ucm/s	ALA3123332		ucm/s	Homo sapiens
15.	ALA3121095	R,S(+)-4a, R,S-4a	PPB	=	77	%	ALA3123330		%
16.	ALA3121095	R,S(+)-4a, R,S-4a	PPB	=	77	%	ALA3123329		%
17.	ALA3121095	R,S(+)-4a, R,S-4a	PPB	=	77	%	ALA3123328		%
18.	ALA3121095	R,S(+)-4a, R,S-4a	solubility	>	1	mg/ml	ALA3123326		ug.mL-1
19.	ALA3121095	R,S(+)-4a, R,S-4a	solubility	=	0.8	mg/ml	ALA3123327		ug.mL-1
20.	ALA3121095	R,S(+)-4a, R,S-4a	beta t1/2	=	2.6	hr	ALA3123325		hr	Rattus norvegicus