| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3122212 | 14, PF470, PF-06297470 | Activity_index | > | 5.4 | ALA4019165 | Mus musculus | |||||
| 2. | ALA3122212 | 14, PF470, PF-06297470 | Ki | = | 0.9 | nM | ALA3124717 | 9.05 | nM | Homo sapiens | ||
| 3. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | = | 2.5 | nM | ALA3124716 | 8.60 | nM | Rattus norvegicus | ||
| 4. | ALA3122212 | 14, PF470, PF-06297470 | CLH | = | 23.7 | ml/min.kg | ALA3124714 | mL.min-1.kg-1 | Homo sapiens | |||
| 5. | ALA3122212 | 14, PF470, PF-06297470 | Ratio IC50 | > | 12000 | ALA3124712 | ||||||
| 6. | ALA3122212 | 14, PF470, PF-06297470 | Papp | = | 22 | ucm/s | ALA3124711 | ucm/s | ||||
| 7. | ALA3122212 | 14, PF470, PF-06297470 | Ratio | = | 1.11 | ALA3124710 | Canis lupus familiaris | |||||
| 8. | ALA3122212 | 14, PF470, PF-06297470 | Fu | = | 0.091 | ALA3124720 | Rattus norvegicus | |||||
| 9. | ALA3122212 | 14, PF470, PF-06297470 | Fu | = | 0.097 | ALA3124721 | Rattus norvegicus | |||||
| 10. | ALA3122212 | 14, PF470, PF-06297470 | t1/2 | = | 0.31 | hr | ALA3124708 | hr | Rattus norvegicus | |||
| 11. | ALA3122212 | 14, PF470, PF-06297470 | F | = | 28 | % | ALA3124707 | % | Rattus norvegicus | |||
| 12. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124706 | nM | Homo sapiens | |||
| 13. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124705 | nM | Homo sapiens | |||
| 14. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124704 | nM | Homo sapiens | |||
| 15. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124703 | nM | Homo sapiens | |||
| 16. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124702 | nM | Homo sapiens | |||
| 17. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124579 | nM | Homo sapiens | |||
| 18. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124578 | nM | Homo sapiens | |||
| 19. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124577 | nM | Homo sapiens | |||
| 20. | ALA3122212 | 14, PF470, PF-06297470 | IC50 | > | 10 | uM | ALA3124576 | nM | Homo sapiens |
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