# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3125459 | 41 | IC50 | = | 2.5 | nM | ALA3130910 | 8.60 | nM | Homo sapiens | ||
2. | ALA3125459 | 41 | IC50 | = | 900 | nM | ALA3130110 | 6.05 | nM | Homo sapiens | ||
3. | ALA3125459 | 41 | Ratio IC50 | = | 360 | ALA3130109 | ||||||
4. | ALA3125459 | 41 | Tmax | = | 1.19 | hr | ALA3130108 | hr | Rattus norvegicus | |||
5. | ALA3125459 | 41 | Cmax | = | 1494 | ng/ml | ALA3130107 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
6. | ALA3125459 | 41 | AUC | = | 7005 | ng.hr/ml | ALA3130106 | ng.hr.mL-1 | Rattus norvegicus | |||
7. | ALA3125459 | 41 | t1/2 | = | 6.34 | hr | ALA3130105 | hr | Rattus norvegicus | |||
8. | ALA3125459 | 41 | Tmax | = | 1.56 | hr | ALA3130104 | hr | Rattus norvegicus | |||
9. | ALA3125459 | 41 | Cmax | = | 257 | ng/ml | ALA3130103 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
10. | ALA3125459 | 41 | AUC | = | 1016 | ng.hr/ml | ALA3130102 | ng.hr.mL-1 | Rattus norvegicus | |||
11. | ALA3125459 | 41 | t1/2 | = | 3.5 | hr | ALA3130101 | hr | Rattus norvegicus | |||
12. | ALA3125459 | 41 | F | = | 76.3 | % | ALA3130100 | % | Rattus norvegicus | |||
13. | ALA3125459 | 41 | AUC | = | 1332 | ng.hr/ml | ALA3130098 | ng.hr.mL-1 | Rattus norvegicus | |||
14. | ALA3125459 | 41 | t1/2 | = | 2.69 | hr | ALA3130099 | hr | Rattus norvegicus | |||
15. | ALA3125459 | 41 | CL | = | 0.76 | L/hr/kg | ALA3130097 | mL.min-1.kg-1 | Rattus norvegicus | |||
16. | ALA3125459 | 41 | Activity | = | 251 | % | ALA3129942 | % | Rattus norvegicus | |||
17. | ALA3125459 | 41 | Activity | = | 1983 | % | ALA3129941 | % | Rattus norvegicus | |||
18. | ALA3125459 | 41 | Activity | = | 2234 | % | ALA3129940 | % | Rattus norvegicus | |||
19. | ALA3125459 | 41 | Activity | = | 3485 | % | ALA3129939 | % | Canis lupus familiaris | |||
20. | ALA3125459 | 41 | Activity | = | 11197 | % | ALA3129938 | % | Canis lupus familiaris |