# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3126396 | 1 | IC50 | > | 1000 | uM | ALA5151872 | nM | Chlorocebus sabaeus | |||
2. | ALA3126396 | 1 | t1/2 | = | 1.7 | hr | ALA5151871 | hr | ||||
3. | ALA3126396 | 1 | Stability | = | 5 | % | ALA5151870 | % | ||||
4. | ALA3126396 | 1 | Ki | = | 19 | nM | ALA5151868 | 7.72 | nM | Homo sapiens | ||
5. | ALA3126396 | 1 | Ki | = | 19 | nM | ALA5151867 | 7.72 | nM | Homo sapiens | ||
6. | ALA3126396 | 1 | t1/2 | = | 3.54 | min | ALA4689554 | hr | ||||
7. | ALA3126396 | 1 | INH | 0 | ALA4689553 | Not Active | % | Homo sapiens | ||||
8. | ALA3126396 | 1 | INH | 0 | ALA4689552 | Active | % | Homo sapiens | ||||
9. | ALA3126396 | 1 | INH | 0 | ALA4689551 | Active | % | Homo sapiens | ||||
10. | ALA3126396 | 1 | Ki | = | 15 | nM | ALA4689550 | 7.82 | nM | Homo sapiens | ||
11. | ALA3126396 | 1 | t1/2 | = | 3.7 | hr | ALA3130018 | hr | Mus musculus | |||
12. | ALA3126396 | 1 | t1/2 | = | 4 | hr | ALA3130021 | hr | ||||
13. | ALA3126396 | 1 | t1/2 | = | 8 | hr | ALA3130020 | hr | Homo sapiens | |||
14. | ALA3126396 | 1 | t1/2 | = | 10 | hr | ALA3130019 | hr | Homo sapiens | |||
15. | ALA3126396 | 1 | Ki | = | 25 | nM | ALA3129874 | 7.60 | nM | Homo sapiens | ||
16. | ALA3126396 | 1 | INH | = | 51 | % | ALA3129873 | % | Homo sapiens | |||
17. | ALA3126396 | 1 | INH | = | 84 | % | ALA3129870 | % | ||||
18. | ALA3126396 | 1 | Activity | < | 5 | % | ALA3129878 | % | ||||
19. | ALA3126396 | 1 | MTD | > | 10 | mg kg-1 | ALA3129875 | mg kg-1 | Mus musculus | |||
20. | ALA3126396 | 1 | IC50 | > | 1000 | uM | ALA3129871 | nM |