| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3127117 | 41 | solubility | = | 45 | uM | ALA3129607 | nM | ||||
| 2. | ALA3127117 | 41 | CLH | = | 18 | microL/min/mg | ALA3129606 | mL.min-1.g-1 | Homo sapiens | |||
| 3. | ALA3127117 | 41 | Papp | = | 6.4 | ucm/s | ALA3129605 | ucm/s | Homo sapiens | |||
| 4. | ALA3127117 | 41 | Papp | = | 74 | ucm/s | ALA3129604 | ucm/s | Homo sapiens | |||
| 5. | ALA3127117 | 41 | Ratio | = | 11.5 | ALA3129603 | Homo sapiens | |||||
| 6. | ALA3127117 | 41 | CL | = | 35 | ml/min.kg | ALA3129602 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA3127117 | 41 | t1/2 | = | 13.2 | hr | ALA3129601 | hr | Rattus norvegicus | |||
| 8. | ALA3127117 | 41 | Vdss | = | 13 | L/Kg | ALA3129600 | L.kg-1 | Rattus norvegicus | |||
| 9. | ALA3127117 | 41 | Cmax | = | 0.08 | uM | ALA3129599 | nM | Rattus norvegicus | |||
| 10. | ALA3127117 | 41 | F | = | 22 | % | ALA3129598 | % | Rattus norvegicus | |||
| 11. | ALA3127117 | 41 | Activity | = | 54 | % | ALA3129597 | % | Rattus norvegicus | |||
| 12. | ALA3127117 | 41 | Activity | = | 55 | % | ALA3129596 | % | Rattus norvegicus | |||
| 13. | ALA3127117 | 41 | pIC50 | = | 8.1 | ALA3129614 | 8.10 | nM | Rattus norvegicus | |||
| 14. | ALA3127117 | 41 | Ratio IC50 | = | 10 | ALA3129592 | ||||||
| 15. | ALA3127117 | 41 | Cp | = | 0.37 | uM | ALA3129594 | uM | Rattus norvegicus | |||
| 16. | ALA3127117 | 41 | pIC50 | = | 9 | ALA3129612 | 9.00 | nM | Homo sapiens |
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