# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3128178 | 19 | Cp(f) | = | 0.09 | uM | ALA3128804 | uM | Rattus norvegicus | |||
2. | ALA3128178 | 19 | Cp(f) | = | 0.26 | uM | ALA3128803 | uM | Rattus norvegicus | |||
3. | ALA3128178 | 19 | Cp(f) | = | 1.17 | uM | ALA3128802 | uM | Rattus norvegicus | |||
4. | ALA3128178 | 19 | EC50 | = | 1.36 | nM | ALA3129374 | 8.87 | nM | Homo sapiens | ||
5. | ALA3128178 | 19 | t1/2 | = | 2 | hr | ALA3129325 | hr | Rattus norvegicus | |||
6. | ALA3128178 | 19 | t1/2 | = | 2 | hr | ALA3129324 | hr | Macaca mulatta | |||
7. | ALA3128178 | 19 | EC50 | = | 2 | nM | ALA3128810 | 8.70 | nM | Macaca mulatta | ||
8. | ALA3128178 | 19 | EC50 | = | 5 | nM | ALA3128845 | 8.30 | nM | Canis lupus familiaris | ||
9. | ALA3128178 | 19 | t1/2 | = | 6 | hr | ALA3129323 | hr | Canis lupus familiaris | |||
10. | ALA3128178 | 19 | IC50 | = | 6.1 | uM | ALA3129316 | 5.21 | nM | Homo sapiens | ||
11. | ALA3128178 | 19 | Fu | = | 19 | % | ALA3129319 | Rattus norvegicus | ||||
12. | ALA3128178 | 19 | Ratio EC50 | = | 20 | ALA3128808 | ||||||
13. | ALA3128178 | 19 | Papp | = | 13 | ucm/s | ALA3129314 | ucm/s | ||||
14. | ALA3128178 | 19 | CL | = | 27 | ml/min.kg | ALA3129326 | mL.min-1.kg-1 | Canis lupus familiaris | |||
15. | ALA3128178 | 19 | EC50 | = | 27.6 | nM | ALA3128847 | 7.56 | nM | Rattus norvegicus | ||
16. | ALA3128178 | 19 | CL | = | 33 | ml/min.kg | ALA3129328 | mL.min-1.kg-1 | Rattus norvegicus | |||
17. | ALA3128178 | 19 | CL | = | 36 | ml/min.kg | ALA3129327 | mL.min-1.kg-1 | Macaca mulatta | |||
18. | ALA3128178 | 19 | F | = | 41 | % | ALA3129322 | % | Rattus norvegicus | |||
19. | ALA3128178 | 19 | F | = | 67 | % | ALA3129320 | % | Canis lupus familiaris | |||
20. | ALA3128178 | 19 | Activity | = | 59 | % | ALA3128805 | % | Rattus norvegicus |