# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3128194 | 11a | EC50 | = | 0.06 | nM | ALA3128810 | 10.22 | nM | Macaca mulatta | ||
2. | ALA3128194 | 11a | EC50 | = | 0.15 | nM | ALA3129374 | 9.82 | nM | Homo sapiens | ||
3. | ALA3128194 | 11a | EC50 | = | 0.19 | nM | ALA3128845 | 9.72 | nM | Canis lupus familiaris | ||
4. | ALA3128194 | 11a | EC50 | = | 1.3 | nM | ALA3128847 | 8.89 | nM | Rattus norvegicus | ||
5. | ALA3128194 | 11a | IC50 | = | 12.7 | uM | ALA3129316 | 4.90 | nM | Homo sapiens | ||
6. | ALA3128194 | 11a | t1/2 | = | 4 | hr | ALA3129325 | hr | Rattus norvegicus | |||
7. | ALA3128194 | 11a | Papp | = | 5 | ucm/s | ALA3129314 | ucm/s | ||||
8. | ALA3128194 | 11a | IC50 | = | 5.6 | uM | ALA3128856 | 5.25 | nM | Homo sapiens | ||
9. | ALA3128194 | 11a | F | = | 6 | % | ALA3129322 | % | Rattus norvegicus | |||
10. | ALA3128194 | 11a | Fu | = | 18 | % | ALA3129319 | Rattus norvegicus | ||||
11. | ALA3128194 | 11a | IC50 | = | 18.3 | uM | ALA3129312 | 4.74 | nM | Homo sapiens | ||
12. | ALA3128194 | 11a | CLH | = | 59 | ml/min.kg | ALA3129315 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA3128194 | 11a | CL | = | 50 | ml/min.kg | ALA3129328 | mL.min-1.kg-1 | Rattus norvegicus | |||
14. | ALA3128194 | 11a | Activity | = | 78 | % | ALA3128809 | % | Macaca mulatta | |||
15. | ALA3128194 | 11a | IC50 | = | 86 | uM | ALA3129311 | 4.07 | nM | Homo sapiens | ||
16. | ALA3128194 | 11a | Activity | = | 91 | % | ALA3129373 | % | Homo sapiens | |||
17. | ALA3128194 | 11a | Activity | = | 100 | % | ALA3128846 | % | Rattus norvegicus | |||
18. | ALA3128194 | 11a | Activity | = | 102 | % | ALA3128844 | % | Canis lupus familiaris | |||
19. | ALA3128194 | 11a | IC50 | = | 1218 | nM | ALA3128855 | 5.91 | nM | Homo sapiens | ||
20. | ALA3128194 | 11a | IC50 | > | 100 | uM | ALA3129313 | nM | Homo sapiens |