# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3142235 | Sitamaquine, WR-6026 | Ratio | 0 | ALA3252345 | Not Active | Trypanosoma cruzi | |||||
2. | ALA3142235 | Sitamaquine, WR-6026 | INH | 0 | ALA3252343 | Not Active | % | Trypanosoma cruzi | ||||
3. | ALA3142235 | Sitamaquine, WR-6026 | INH | 0 | ALA3252342 | Not Active | % | Trypanosoma cruzi | ||||
4. | ALA3142235 | Sitamaquine, WR-6026 | INH | 0 | ALA3252341 | Not Active | % | Trypanosoma cruzi | ||||
5. | ALA3142235 | Sitamaquine, WR-6026 | Ratio EC50 | = | 2 | ALA1692847 | Leishmania major | |||||
6. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 24.49 | uM | ALA1692848 | 4.61 | nM | Leishmania major | ||
7. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 12.02 | uM | ALA1692849 | 4.92 | nM | Leishmania major | ||
8. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679119 | Active | Leishmania tropica | |||||
9. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679118 | Active | Leishmania tropica | |||||
10. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679117 | Active | Leishmania donovani | |||||
11. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679116 | Active | Leishmania donovani | |||||
12. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679115 | Not Active | Leishmania donovani | |||||
13. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679114 | Not Active | Leishmania donovani | |||||
14. | ALA3142235 | Sitamaquine, WR-6026 | Drug uptake | 0 | ALA1679113 | Not Active | Leishmania donovani | |||||
15. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 5.7 | uM | ALA1678993 | 5.24 | nM | Leishmania sp. | ||
16. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 9.5 | uM | ALA1681020 | 5.02 | nM | Leishmania tropica | ||
17. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 9.5 | uM | ALA1681019 | 5.02 | nM | Leishmania braziliensis | ||
18. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 9.5 | uM | ALA1681018 | 5.02 | nM | Leishmania mexicana | ||
19. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 9.5 | uM | ALA1681017 | 5.02 | nM | Leishmania infantum | ||
20. | ALA3142235 | Sitamaquine, WR-6026 | EC50 | = | 9.5 | uM | ALA1681016 | 5.02 | nM | Leishmania donovani |