| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA327721 | 3f | IC50 | = | 16 | nM | ALA5138021 | 7.80 | nM | Homo sapiens | ||
| 2. | ALA327721 | 3f | Activity | = | 16 | nM | ALA969299 | nM | Homo sapiens | |||
| 3. | ALA327721 | 3f | IC50 | = | 328 | nM | ALA690693 | 6.48 | nM | Homo sapiens | ||
| 4. | ALA327721 | 3f | Solubility | > | 0.205 | mg mL-1 | ALA633684 | ug.mL-1 | ||||
| 5. | ALA327721 | 3f | Solubility | = | 18.17 | mg mL-1 | ALA634516 | ug.mL-1 | ||||
| 6. | ALA327721 | 3f | logP | = | 3.7 | ALA630087 | ||||||
| 7. | ALA327721 | 3f | Selectivity | = | 147 | ALA843964 | Homo sapiens | |||||
| 8. | ALA327721 | 3f | Selectivity | = | 136 | ALA843960 | Homo sapiens | |||||
| 9. | ALA327721 | 3f | Selectivity | = | 246 | ALA843959 | Homo sapiens | |||||
| 10. | ALA327721 | 3f | Selectivity | = | 3 | ALA843962 | Homo sapiens | |||||
| 11. | ALA327721 | 3f | Selectivity | = | 20 | ALA843961 | Homo sapiens | |||||
| 12. | ALA327721 | 3f | Selectivity | = | 7 | ALA843963 | Homo sapiens | |||||
| 13. | ALA327721 | 3f | F | = | 33 | % | ALA618792 | % | Rattus norvegicus | |||
| 14. | ALA327721 | 3f | Vdss | = | 1.7 | l kg-1 | ALA618527 | L.kg-1 | Rattus norvegicus | |||
| 15. | ALA327721 | 3f | T1/2 | = | 1.8 | hr | ALA625865 | hr | Rattus norvegicus | |||
| 16. | ALA327721 | 3f | Cl | = | 13 | ml min-1 kg-1 | ALA621796 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA327721 | 3f | IC50 | = | 16 | nM | ALA819548 | 7.80 | nM | Homo sapiens |
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