| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3234871 | 45h | Activity | 0 | ALA3239484 | Active | Mus musculus | |||||
| 2. | ALA3234871 | 45h | Activity | > | 10 | uM | ALA3239447 | uM | Homo sapiens | |||
| 3. | ALA3234871 | 45h | FC | = | 3.9 | ALA3239497 | Mus musculus | |||||
| 4. | ALA3234871 | 45h | FC | = | 4.1 | ALA3239496 | Mus musculus | |||||
| 5. | ALA3234871 | 45h | Efficacy | = | 100 | % | ALA3239495 | % | Mus musculus | |||
| 6. | ALA3234871 | 45h | Efficacy | = | 100 | % | ALA3239494 | % | Homo sapiens | |||
| 7. | ALA3234871 | 45h | Ratio AUC | = | 0.8 | ALA3239489 | Mus musculus | |||||
| 8. | ALA3234871 | 45h | AUC | = | 37452 | nM.hr | ALA3239488 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 9. | ALA3234871 | 45h | AUC | = | 45469 | nM.hr | ALA3239487 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 10. | ALA3234871 | 45h | Cmax | = | 5165 | nM | ALA3239486 | nM | Mus musculus | |||
| 11. | ALA3234871 | 45h | Cmax | = | 4770 | nM | ALA3239485 | nM | Mus musculus | |||
| 12. | ALA3234871 | 45h | FC | = | 3.1 | ALA3239451 | Mus musculus | |||||
| 13. | ALA3234871 | 45h | INH | = | 4.6 | uM | ALA3239450 | uM | Homo sapiens | |||
| 14. | ALA3234871 | 45h | PPB | = | 99.9 | % | ALA3239449 | % | ||||
| 15. | ALA3234871 | 45h | logD | = | 2.5 | ALA3239448 | ||||||
| 16. | ALA3234871 | 45h | AUC | = | 11393 | nM.hr | ALA3239446 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 17. | ALA3234871 | 45h | F | = | 96.5 | % | ALA3239442 | % | Mus musculus | |||
| 18. | ALA3234871 | 45h | t1/2 | = | 11.7 | hr | ALA3239441 | hr | Mus musculus | |||
| 19. | ALA3234871 | 45h | t1/2 | = | 4.14 | hr | ALA3239440 | hr | Mus musculus | |||
| 20. | ALA3234871 | 45h | Cmax | = | 9750 | nM | ALA3239439 | nM | Mus musculus |
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