# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3235419 | 8, BDM43124 | Papp | = | 0.2 | ucm/s | ALA3243756 | ucm/s | Homo sapiens | |||
2. | ALA3235419 | 8, BDM43124 | Activity | = | 62 | % | ALA3239896 | % | Homo sapiens | |||
3. | ALA3235419 | 8, BDM43124 | Activity | = | 132.5 | ug/L | ALA3239895 | ug/L | Mus musculus | |||
4. | ALA3235419 | 8, BDM43124 | Activity | = | 78.8 | ug/L | ALA3239894 | ug/L | Mus musculus | |||
5. | ALA3235419 | 8, BDM43124 | Activity | = | 21.2 | ug/L | ALA3239893 | ug/L | Mus musculus | |||
6. | ALA3235419 | 8, BDM43124 | INH | 0 | ALA3239892 | Not Active | % | Homo sapiens | ||||
7. | ALA3235419 | 8, BDM43124 | INH | 0 | ALA3239891 | Not Active | % | Homo sapiens | ||||
8. | ALA3235419 | 8, BDM43124 | INH | 0 | ALA3239890 | Dose-dependent effect | % | Homo sapiens | ||||
9. | ALA3235419 | 8, BDM43124 | INH | 0 | ALA3243762 | Dose-dependent effect | % | Homo sapiens | ||||
10. | ALA3235419 | 8, BDM43124 | t1/2 | = | 11.3 | hr | ALA3243758 | hr | ||||
11. | ALA3235419 | 8, BDM43124 | t1/2 | = | 0.1 | hr | ALA3243757 | hr | Mus musculus | |||
12. | ALA3235419 | 8, BDM43124 | logD | = | 1.1 | ALA3243755 | ||||||
13. | ALA3235419 | 8, BDM43124 | solubility | = | 74 | uM | ALA3243754 | nM | ||||
14. | ALA3235419 | 8, BDM43124 | Activity | = | 50 | % | ALA3243753 | % | Homo sapiens | |||
15. | ALA3235419 | 8, BDM43124 | IC50 | > | 100 | uM | ALA3243737 | nM | Homo sapiens |