| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3261926 | 10 | t1/2 | = | 0.36 | hr | ALA4813589 | hr | ||||
| 2. | ALA3261926 | 10 | Stabilty | = | 15 | % | ALA4813586 | % | ||||
| 3. | ALA3261926 | 10 | IC50 | = | 5 | nM | ALA4813584 | 8.30 | nM | Homo sapiens | ||
| 4. | ALA3261926 | 10 | IC50 | = | 1 | nM | ALA4813583 | 9.00 | nM | Homo sapiens | ||
| 5. | ALA3261926 | 10 | INH | = | 99.9 | % | ALA4813582 | % | Homo sapiens | |||
| 6. | ALA3261926 | 10 | INH | = | 99.2 | % | ALA4813581 | % | Homo sapiens | |||
| 7. | ALA3261926 | 10 | IC50 | = | 2.9 | nM | ALA4398559 | 8.54 | nM | Homo sapiens | ||
| 8. | ALA3261926 | 10 | Activity | 0 | ALA4398558 | Active | Mus musculus | |||||
| 9. | ALA3261926 | 10 | Activity | 0 | ALA4398557 | Active | Mus musculus | |||||
| 10. | ALA3261926 | 10 | pIC50 | = | 9.1 | ALA3859628 | 9.10 | nM | Homo sapiens | |||
| 11. | ALA3261926 | 10 | pIC50 | = | 8.1 | ALA3859629 | 8.10 | nM | Homo sapiens | |||
| 12. | ALA3261926 | 10 | t1/2 | < | 1 | hr | ALA3859630 | hr | ||||
| 13. | ALA3261926 | 10 | pIC50 | < | 5 | ALA3268203 | nM | Homo sapiens | ||||
| 14. | ALA3261926 | 10 | pIC50 | < | 5 | ALA3268206 | nM | Homo sapiens | ||||
| 15. | ALA3261926 | 10 | pIC50 | < | 5 | ALA3268205 | nM | Homo sapiens | ||||
| 16. | ALA3261926 | 10 | pIC50 | < | 5 | ALA3268204 | nM | Homo sapiens | ||||
| 17. | ALA3261926 | 10 | F | = | 92 | % | ALA3266713 | % | Rattus norvegicus | |||
| 18. | ALA3261926 | 10 | t1/2 | = | 3.5 | hr | ALA3266712 | hr | Rattus norvegicus | |||
| 19. | ALA3261926 | 10 | Vdss | = | 1.9 | L/Kg | ALA3266711 | L.kg-1 | Rattus norvegicus | |||
| 20. | ALA3261926 | 10 | CL | = | 9 | ml/min.kg | ALA3266710 | mL.min-1.kg-1 | Rattus norvegicus |
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