| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3262727 | 12 | IC50 | = | 4.13 | uM | ALA5253347 | 5.38 | nM | Homo sapiens | ||
| 2. | ALA3262727 | 12 | IC50 | = | 5.34 | uM | ALA5253345 | 5.27 | nM | Homo sapiens | ||
| 3. | ALA3262727 | 12 | IC50 | = | 1.39 | uM | ALA5253344 | 5.86 | nM | Homo sapiens | ||
| 4. | ALA3262727 | 12 | IC50 | = | 4.11 | uM | ALA5253343 | 5.39 | nM | Homo sapiens | ||
| 5. | ALA3262727 | 12 | IC50 | = | 0.005 | uM | ALA5253342 | 8.28 | nM | Homo sapiens | ||
| 6. | ALA3262727 | 12 | IC50 | = | 8.73 | uM | ALA5253341 | 5.06 | nM | Homo sapiens | ||
| 7. | ALA3262727 | 12 | IC50 | = | 1.16 | uM | ALA5253338 | 5.94 | nM | Homo sapiens | ||
| 8. | ALA3262727 | 12 | IC50 | = | 0.31 | uM | ALA5253337 | 6.51 | nM | Homo sapiens | ||
| 9. | ALA3262727 | 12 | Ratio IC50 | = | 223 | ALA3266030 | ||||||
| 10. | ALA3262727 | 12 | Ratio IC50 | = | 60 | ALA3266029 | ||||||
| 11. | ALA3262727 | 12 | IC50 | = | 0.005 | uM | ALA3265665 | 8.28 | nM | Homo sapiens | ||
| 12. | ALA3262727 | 12 | IC50 | = | 1.16 | uM | ALA3265664 | 5.94 | nM | Homo sapiens | ||
| 13. | ALA3262727 | 12 | IC50 | = | 0.31 | uM | ALA3265663 | 6.51 | nM | Homo sapiens | ||
| 14. | ALA3262727 | 12 | F | = | 33 | % | ALA3266048 | % | Mus musculus | |||
| 15. | ALA3262727 | 12 | Tmax | = | 0.3 | hr | ALA3266047 | hr | Mus musculus | |||
| 16. | ALA3262727 | 12 | Cmax | = | 409 | ng/ml | ALA3266046 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 17. | ALA3262727 | 12 | t1/2 | = | 2.4 | hr | ALA3266045 | hr | Mus musculus | |||
| 18. | ALA3262727 | 12 | AUC | = | 466 | ng/mL.hr | ALA3266044 | ng.hr.mL-1 | Mus musculus | |||
| 19. | ALA3262727 | 12 | Vdss | = | 9.8 | L/Kg | ALA3266043 | L.kg-1 | Mus musculus | |||
| 20. | ALA3262727 | 12 | CL | = | 127 | ml/min.kg | ALA3266042 | mL.min-1.kg-1 | Mus musculus |
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