| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1137 | 1c | Fu | = | 0.26 | ALA3529402 | ||||||
| 2. | ALA1137 | 1c | CL | = | 66 | ml/min.kg | ALA3529403 | mL.min-1.kg-1 | Homo sapiens | |||
| 3. | ALA1137 | 1c | CL free | = | 5 | ml/min.kg | ALA3529401 | mL.min-1.kg-1 | Homo sapiens | |||
| 4. | ALA1137 | 1c | CL free | = | 248 | ml/min.kg | ALA3529400 | mL.min-1.kg-1 | Homo sapiens | |||
| 5. | ALA1137 | 1c | logP | = | 0.39 | ALA3252779 | ||||||
| 6. | ALA1137 | 1c | Selectivity Index | = | 1.8 | ALA3252778 | ||||||
| 7. | ALA1137 | 1c | pED40 | = | 4.39 | ALA3252776 | ||||||
| 8. | ALA1137 | 1c | pED40 | = | 4.6 | ALA3252774 | Oryctolagus cuniculus | |||||
| 9. | ALA1137 | 1c | Relative potency | = | 0.13 | ALA667670 | Canis lupus familiaris | |||||
| 10. | ALA1137 | 1c | Relative potency | = | 0.77 | ALA646925 | ||||||
| 11. | ALA1137 | 1c | logD | = | 0.53 | ALA635959 | ||||||
| 12. | ALA1137 | 1c | Dose | = | 4.35 | mg | ALA668577 | mg | Canis lupus familiaris | |||
| 13. | ALA1137 | 1c | pA2 app | = | 7.5 | ALA879852 | 7.50 | nM | Canis lupus familiaris | |||
| 14. | ALA1137 | 1c | pA2 app | = | 7.54 | ALA668341 | 7.54 | nM | Canis lupus familiaris | |||
| 15. | ALA1137 | 1c | pA2 app | = | 7.34 | ALA668342 | 7.34 | nM | Canis lupus familiaris | |||
| 16. | ALA1137 | 1c | pA2 | = | 8.62 | ALA652296 | 8.62 | nM | Canis lupus familiaris | |||
| 17. | ALA1137 | 1c | pA2 | = | 8.24 | ALA655647 | 8.24 | nM | Cavia porcellus | |||
| 18. | ALA1137 | 1c | Vasodilation | = | 4.82 | ALA649671 | Canis lupus familiaris | |||||
| 19. | ALA1137 | 1c | Contractile force | = | 4.75 | ALA654265 | Homo sapiens | |||||
| 20. | ALA1137 | 1c | Heart rate | = | 5.12 | ALA647666 | Homo sapiens |
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