| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3263691 | 9j | Selectivity ratio | > | 1000 | ALA3270931 | ||||||
| 2. | ALA3263691 | 9j | Selectivity ratio | > | 1000 | ALA3270930 | ||||||
| 3. | ALA3263691 | 9j | solubility | = | 160 | uM | ALA3270929 | nM | ||||
| 4. | ALA3263691 | 9j | Vdss | = | 5.46 | L/Kg | ALA3270928 | L.kg-1 | Rattus norvegicus | |||
| 5. | ALA3263691 | 9j | CL | = | 13.2 | ml/min.kg | ALA3270927 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA3263691 | 9j | F | = | 21 | % | ALA3270557 | % | Rattus norvegicus | |||
| 7. | ALA3263691 | 9j | Efficacy | = | 78 | % | ALA3270926 | % | ||||
| 8. | ALA3263691 | 9j | EC50 | = | 170 | nM | ALA3270563 | 6.77 | nM | |||
| 9. | ALA3263691 | 9j | CL | = | 18 | microL/min/mg | ALA3270561 | mL.min-1.g-1 | ||||
| 10. | ALA3263691 | 9j | CL | = | 20 | microL/min/mg | ALA3270562 | mL.min-1.g-1 | ||||
| 11. | ALA3263691 | 9j | EC50 | = | 89 | uM | ALA3270558 | 4.05 | nM | Homo sapiens | ||
| 12. | ALA3263691 | 9j | EC50 | = | 0.1 | uM | ALA3812619 | 7.00 | nM | Homo sapiens | ||
| 13. | ALA3263691 | 9j | EC50 | < | 0.1 | uM | ALA3812618 | nM | Homo sapiens |
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