| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3286660 | 7z, TG8-15 | solubility | = | 500 | uM | ALA5224048 | nM | ||||
| 2. | ALA3286660 | 7z, TG8-15 | BPR | = | 0.02 | ALA5224047 | ||||||
| 3. | ALA3286660 | 7z, TG8-15 | t1/2 | = | 10.5 | hr | ALA5224046 | hr | ||||
| 4. | ALA3286660 | 7z, TG8-15 | Kb | = | 130 | uM | ALA5224045 | nM | Homo sapiens | |||
| 5. | ALA3286660 | 7z, TG8-15 | Kb | = | 15 | uM | ALA5224044 | nM | Homo sapiens | |||
| 6. | ALA3286660 | 7z, TG8-15 | Kb | = | 18 | uM | ALA5224043 | nM | Homo sapiens | |||
| 7. | ALA3286660 | 7z, TG8-15 | Kb | = | 48.5 | nM | ALA5224042 | nM | Homo sapiens | |||
| 8. | ALA3286660 | 7z, TG8-15 | KB | = | 22.2 | nM | ALA5121386 | nM | Homo sapiens | |||
| 9. | ALA3286660 | 7z, TG8-15 | Therm_solubility | = | 257 | nM | ALA5121331 | nM | ||||
| 10. | ALA3286660 | 7z, TG8-15 | AUC | = | 156 | nM | ALA3293439 | nM | Mus musculus | |||
| 11. | ALA3286660 | 7z, TG8-15 | AUClast | = | 125 | nM | ALA3293438 | nM | Mus musculus | |||
| 12. | ALA3286660 | 7z, TG8-15 | Cmax | = | 134 | nM | ALA3293437 | nM | Mus musculus | |||
| 13. | ALA3286660 | 7z, TG8-15 | beta t1/2 | = | 0.3 | hr | ALA3293436 | hr | Mus musculus | |||
| 14. | ALA3286660 | 7z, TG8-15 | AUC | = | 1600 | hr.ng/ml | ALA3293435 | ng.hr.mL-1 | Mus musculus | |||
| 15. | ALA3286660 | 7z, TG8-15 | AUClast | = | 1580 | hr.ng/ml | ALA3293434 | ng.hr.mL-1 | Mus musculus | |||
| 16. | ALA3286660 | 7z, TG8-15 | Cmax | = | 2040 | ng/ml | ALA3293433 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 17. | ALA3286660 | 7z, TG8-15 | solubility | = | 257 | uM | ALA3293432 | nM | ||||
| 18. | ALA3286660 | 7z, TG8-15 | Stability | = | 57 | % | ALA3293431 | % | Mus musculus | |||
| 19. | ALA3286660 | 7z, TG8-15 | Stability | = | 75 | % | ALA3293430 | % | Mus musculus | |||
| 20. | ALA3286660 | 7z, TG8-15 | Stability | = | 85 | % | ALA3293429 | % | Mus musculus |
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