| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3287695 | 44 | Tmax | = | 30 | hr | ALA3294097 | hr | Rattus norvegicus | |||
| 2. | ALA3287695 | 44 | Emax | = | 83.3 | % | ALA3294096 | % | Rattus norvegicus | |||
| 3. | ALA3287695 | 44 | Ratio | = | 18 | ALA3294095 | ||||||
| 4. | ALA3287695 | 44 | BPR | = | 0.03 | ALA3294087 | ||||||
| 5. | ALA3287695 | 44 | Drug uptake | = | 0.23 | uM | ALA3294086 | uM | Rattus norvegicus | |||
| 6. | ALA3287695 | 44 | beta t1/2 | = | 43 | min | ALA3294085 | hr | Rattus norvegicus | |||
| 7. | ALA3287695 | 44 | Cp | = | 10.57 | uM | ALA3294084 | uM | Rattus norvegicus | |||
| 8. | ALA3287695 | 44 | Emax | = | 91.2 | % | ALA3294083 | % | Rattus norvegicus | |||
| 9. | ALA3287695 | 44 | EC50 | = | 12 | nM | ALA3294082 | 7.92 | nM | Rattus norvegicus | ||
| 10. | ALA3287695 | 44 | Emax | = | 78.2 | % | ALA3294081 | % | Rattus norvegicus | |||
| 11. | ALA3287695 | 44 | EC50 | = | 1771 | nM | ALA3294080 | 5.75 | nM | Rattus norvegicus | ||
| 12. | ALA3287695 | 44 | FC | = | 5.48 | ALA3294079 | Rattus norvegicus | |||||
| 13. | ALA3287695 | 44 | FC | = | 4.5 | ALA3291875 | Rattus norvegicus | |||||
| 14. | ALA3287695 | 44 | Activity | 0 | ALA3291874 | Dose-dependent effect | Rattus norvegicus | |||||
| 15. | ALA3287695 | 44 | Activity | 0 | ALA3291873 | Dose-dependent effect | Rattus norvegicus | |||||
| 16. | ALA3287695 | 44 | Activity | 0 | ALA3291871 | Not Active | Rattus norvegicus | |||||
| 17. | ALA3287695 | 44 | EC50 | = | 148 | nM | ALA3291872 | 6.83 | nM | Rattus norvegicus | ||
| 18. | ALA3287695 | 44 | beta t1/2 | = | 28 | min | ALA3291870 | hr | Rattus norvegicus | |||
| 19. | ALA3287695 | 44 | AUCt | = | 304.6 | umol.min/L | ALA3291869 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 20. | ALA3287695 | 44 | Vdss | = | 0.55 | L/Kg | ALA3291868 | L.kg-1 | Rattus norvegicus |
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