| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3288029 | 12a | ED80 | = | 0.2 | ug/kg | ALA3295487 | ug/kg | Rattus norvegicus | |||
| 2. | ALA3288029 | 12a | ED80 | = | 23 | nM | ALA3295486 | nM | Rattus norvegicus | |||
| 3. | ALA3288029 | 12a | Activity | = | 90 | nM | ALA3295492 | nM | Rattus norvegicus | |||
| 4. | ALA3288029 | 12a | Activity | = | 30 | nM | ALA3295491 | nM | Rattus norvegicus | |||
| 5. | ALA3288029 | 12a | Activity | = | 12 | nM | ALA3295490 | nM | Rattus norvegicus | |||
| 6. | ALA3288029 | 12a | Activity | = | 2 | nM | ALA3295489 | nM | Rattus norvegicus | |||
| 7. | ALA3288029 | 12a | t1/2 | = | 15 | hr | ALA3295485 | hr | Canis lupus familiaris | |||
| 8. | ALA3288029 | 12a | F | = | 16 | % | ALA3295484 | % | Canis lupus familiaris | |||
| 9. | ALA3288029 | 12a | Vz/F | = | 44 | L/Kg | ALA3295483 | L.kg-1 | Canis lupus familiaris | |||
| 10. | ALA3288029 | 12a | Vdss | = | 26 | L/Kg | ALA3295228 | L.kg-1 | Canis lupus familiaris | |||
| 11. | ALA3288029 | 12a | CL | = | 34 | ml/min.kg | ALA3292513 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 12. | ALA3288029 | 12a | pIC50 | = | 4.7 | ALA3292514 | 4.70 | nM | Homo sapiens | |||
| 13. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3292517 | ||||||
| 14. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3292516 | ||||||
| 15. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3292519 | ||||||
| 16. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3292518 | ||||||
| 17. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3295227 | ||||||
| 18. | ALA3288029 | 12a | Selectivity ratio | > | 10000 | ALA3295226 | ||||||
| 19. | ALA3288029 | 12a | pIC50 | = | 10.7 | ALA3295225 | 10.70 | nM | Rattus norvegicus | |||
| 20. | ALA3288029 | 12a | pIC50 | > | 8 | ALA3295224 | nM | Homo sapiens |
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