| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3290657 | 20 | Activity | 0 | ALA3294651 | Dose-dependent effect | Rattus norvegicus | |||||
| 2. | ALA3290657 | 20 | Activity | 0 | ALA3294650 | Dose-dependent effect | Rattus norvegicus | |||||
| 3. | ALA3290657 | 20 | Activity | 0 | ALA3294649 | Not Active | Homo sapiens | |||||
| 4. | ALA3290657 | 20 | Activity | 0 | ALA3294648 | Not Active | Homo sapiens | |||||
| 5. | ALA3290657 | 20 | solubility | > | 200 | uM/ml | ALA3294647 | nM | ||||
| 6. | ALA3290657 | 20 | PPB | < | 0.1 | % | ALA3294646 | % | ||||
| 7. | ALA3290657 | 20 | PPB | < | 0.1 | % | ALA3294645 | % | ||||
| 8. | ALA3290657 | 20 | F | > | 99 | % | ALA3294644 | % | Canis lupus familiaris | |||
| 9. | ALA3290657 | 20 | F | = | 86 | % | ALA3294643 | % | Rattus norvegicus | |||
| 10. | ALA3290657 | 20 | t1/2 | = | 3.6 | hr | ALA3294642 | hr | Canis lupus familiaris | |||
| 11. | ALA3290657 | 20 | t1/2 | = | 0.9 | hr | ALA3294641 | hr | Rattus norvegicus | |||
| 12. | ALA3290657 | 20 | CL | = | 9.6 | ml/min.kg | ALA3294640 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 13. | ALA3290657 | 20 | CL | = | 21 | ml/min.kg | ALA3294639 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA3290657 | 20 | IC50 | = | 1.3 | nM | ALA3294636 | 8.89 | nM | Homo sapiens | ||
| 15. | ALA3290657 | 20 | IC50 | = | 40 | nM | ALA3294635 | 7.40 | nM | Homo sapiens |
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