# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3291427 | 22 | permeability | = | 31 | ucm/s | ALA3292149 | ucm/s | Homo sapiens | |||
2. | ALA3291427 | 22 | solubility | = | 315 | uM | ALA3292123 | nM | ||||
3. | ALA3291427 | 22 | t1/2 | = | 2 | hr | ALA3292146 | hr | Mus musculus | |||
4. | ALA3291427 | 22 | AUC | = | 286 | uM.hr | ALA3292143 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
5. | ALA3291427 | 22 | Tmax | = | 0.5 | hr | ALA3292140 | hr | Mus musculus | |||
6. | ALA3291427 | 22 | Cmax | = | 105 | uM | ALA3292137 | nM | Mus musculus | |||
7. | ALA3291427 | 22 | F | = | 100 | % | ALA3292133 | % | Rattus norvegicus | |||
8. | ALA3291427 | 22 | CL | = | 12 | ml/min.kg | ALA3292132 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA3291427 | 22 | IC50 | > | 33 | uM | ALA3292131 | nM | Homo sapiens | |||
10. | ALA3291427 | 22 | IC50 | > | 50 | uM | ALA3292130 | nM | Homo sapiens | |||
11. | ALA3291427 | 22 | IC50 | > | 50 | uM | ALA3292129 | nM | Homo sapiens | |||
12. | ALA3291427 | 22 | IC50 | > | 50 | uM | ALA3292128 | nM | Homo sapiens | |||
13. | ALA3291427 | 22 | IC50 | > | 50 | uM | ALA3292127 | nM | Homo sapiens | |||
14. | ALA3291427 | 22 | IC50 | > | 50 | uM | ALA3292126 | nM | Homo sapiens | |||
15. | ALA3291427 | 22 | permeability | = | 11 | ucm/s | ALA3292125 | ucm/s | Homo sapiens | |||
16. | ALA3291427 | 22 | Fu | = | 17 | % | ALA3292124 | Homo sapiens | ||||
17. | ALA3291427 | 22 | IC50 | = | 2 | uM | ALA3291855 | 5.70 | nM | Homo sapiens | ||
18. | ALA3291427 | 22 | logD | = | 1.6 | ALA3291857 | ||||||
19. | ALA3291427 | 22 | CLH | < | 24 | microL/min/mg | ALA3291856 | mL.min-1.g-1 | Mus musculus | |||
20. | ALA3291427 | 22 | IC50 | = | 0.019 | uM | ALA3291854 | 7.72 | nM |