| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3298242 | 17 | F | = | 37 | % | ALA3299574 | % | Rattus norvegicus | |||
| 2. | ALA3298242 | 17 | Tmax | = | 0.5 | hr | ALA3299573 | hr | Rattus norvegicus | |||
| 3. | ALA3298242 | 17 | Cmax | = | 4769 | nM | ALA3299572 | nM | Rattus norvegicus | |||
| 4. | ALA3298242 | 17 | AUC | = | 15736 | hr.nM | ALA3299571 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA3298242 | 17 | t1/2 | = | 3.5 | hr | ALA3299568 | hr | Rattus norvegicus | |||
| 6. | ALA3298242 | 17 | Vdss | = | 2.06 | L/Kg | ALA3299565 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA3298242 | 17 | CL | = | 14.7 | ml/min.kg | ALA3299562 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA3298242 | 17 | INH | = | 100 | % | ALA3299561 | % | Homo sapiens | |||
| 9. | ALA3298242 | 17 | IC50 | = | 0.55 | uM | ALA3299561 | 6.26 | nM | Homo sapiens | ||
| 10. | ALA3298242 | 17 | INH | = | 97 | % | ALA3299560 | % | Homo sapiens | |||
| 11. | ALA3298242 | 17 | IC50 | = | 0.084 | uM | ALA3299560 | 7.08 | nM | Homo sapiens | ||
| 12. | ALA3298242 | 17 | Ratio IC50 | > | 100 | ALA3299559 | ||||||
| 13. | ALA3298242 | 17 | Ratio IC50 | > | 100 | ALA3299558 | ||||||
| 14. | ALA3298242 | 17 | Ratio IC50 | > | 100 | ALA3299557 | ||||||
| 15. | ALA3298242 | 17 | INH | = | 95 | % | ALA3299556 | % | Homo sapiens | |||
| 16. | ALA3298242 | 17 | IC50 | = | 9 | uM | ALA3299556 | 5.05 | nM | Homo sapiens | ||
| 17. | ALA3298242 | 17 | IC50 | > | 30 | uM | ALA3299555 | nM | Homo sapiens | |||
| 18. | ALA3298242 | 17 | INH | = | 10 | % | ALA3299555 | % | Homo sapiens | |||
| 19. | ALA3298242 | 17 | IC50 | > | 30 | uM | ALA3299554 | nM | Homo sapiens | |||
| 20. | ALA3298242 | 17 | INH | = | 34 | % | ALA3299554 | % | Homo sapiens |
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