# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3298371 | 28 | Ratio IC50 | = | 85 | ALA3428428 | ||||||
2. | ALA3298371 | 28 | Activity | = | 88 | % | ALA3429293 | % | ||||
3. | ALA3298371 | 28 | Activity | = | 102 | % | ALA3429292 | % | Homo sapiens | |||
4. | ALA3298371 | 28 | Activity | = | 96 | % | ALA3429291 | % | Homo sapiens | |||
5. | ALA3298371 | 28 | Activity | = | 96 | % | ALA3429290 | % | Homo sapiens | |||
6. | ALA3298371 | 28 | Activity | = | 96 | % | ALA3429289 | % | Homo sapiens | |||
7. | ALA3298371 | 28 | IC50 | = | 6.2 | uM | ALA3428434 | 5.21 | nM | |||
8. | ALA3298371 | 28 | INH | = | 88 | % | ALA3428433 | % | Homo sapiens | |||
9. | ALA3298371 | 28 | Ratio Ki | = | 470 | ALA3428426 | ||||||
10. | ALA3298371 | 28 | Ki | = | 0.34 | uM | ALA3428283 | 6.47 | nM | Homo sapiens | ||
11. | ALA3298371 | 28 | IC50 | = | 0.045 | uM | ALA3428281 | 7.35 | nM | Homo sapiens | ||
12. | ALA3298371 | 28 | IC50 | = | 4.7 | uM | ALA3428282 | 5.33 | nM | |||
13. | ALA3298371 | 28 | INH | = | 98 | % | ALA3371448 | % | Homo sapiens | |||
14. | ALA3298371 | 28 | Ratio Ki | = | 660 | ALA3380551 | ||||||
15. | ALA3298371 | 28 | Ki | = | 460 | nM | ALA3380550 | 6.34 | nM | Homo sapiens | ||
16. | ALA3298371 | 28 | F | = | 100 | % | ALA3371447 | % | Canis lupus familiaris | |||
17. | ALA3298371 | 28 | PPB | = | 93 | % | ALA3371426 | % | ||||
18. | ALA3298371 | 28 | CL | = | 70 | ml/min.kg | ALA3371437 | mL.min-1.kg-1 | Rattus norvegicus | |||
19. | ALA3298371 | 28 | Kinetic_solubility | = | 68 | uM | ALA3380552 | nM | ||||
20. | ALA3298371 | 28 | IC50 | = | 55 | nM | ALA3380549 | 7.26 | nM | Homo sapiens |