# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA321208 | 4b | Inhibition | = | 1 | uM | ALA845618 | uM | ||||
2. | ALA321208 | 4b | Enhancement | = | 0.1 | uM | ALA849952 | uM | ||||
3. | ALA321208 | 4b | IC50 | = | 2.9 | nM | ALA662771 | 8.54 | nM | Cricetulus griseus | ||
4. | ALA321208 | 4b | IC50 | = | 1.2 | nM | ALA620367 | 8.92 | nM | Homo sapiens | ||
5. | ALA321208 | 4b | IC50 | = | 0.12 | nM | ALA880164 | 9.92 | nM | Homo sapiens | ||
6. | ALA321208 | 4b | Lactone | = | 59.4 | % | ALA644888 | % | ||||
7. | ALA321208 | 4b | Lactone | = | 12.2 | % | ALA644886 | % | ||||
8. | ALA321208 | 4b | Lactone | = | 0.1 | % | ALA644887 | % | ||||
9. | ALA321208 | 4b | Lactone | = | 1 | % | ALA644889 | % | Homo sapiens | |||
10. | ALA321208 | 4b | T1/2 | = | 79.4 | min | ALA638883 | hr | ||||
11. | ALA321208 | 4b | T1/2 | = | 27.9 | min | ALA636134 | hr | ||||
12. | ALA321208 | 4b | T1/2 | = | 46.3 | min | ALA636135 | hr | ||||
13. | ALA321208 | 4b | T1/2 | = | 71 | min | ALA636133 | hr | Homo sapiens | |||
14. | ALA321208 | 4b | KDMPC | = | 16000 | M-1 | ALA637327 | M-1 | ||||
15. | ALA321208 | 4b | KDMPC | = | 15500 | M-1 | ALA630139 | M-1 |